P7. Catalytic enantioselective 6𝝿 photocyclization of acrylanilides.
Jones, B., Solon, P., Popescu, M., Du, J.-Y., Paton, R. and Smith, M. D.
ChemRxiv, 2022, Preprint.

P6. Blue light-activatable DNA for remote control of cell-free logic gates and synthetic cells.
Hartmann, D., Chowdhry, R., Smith, J. and Booth, M.
ChemRxiv, 2022, Preprint.

P5. Control of stereogenic oxygen in a helically chiral oxonium ion.
Smith, O., Popescu, M., Hindson, M., Paton, R., Burton, J. and Smith, M. D.
ChemRxiv, 2022, Preprint.

P4. Engineering cellular communication between light-activated synthetic cells and bacteria.
Smith, J. M., Hartmann, D. and Booth, M. J.
bioRxiv, 2022, Preprint.

P3. Catalytic Enantioselective Nucleophilic Desymmetrisation of Phosphonate Esters.
Formica, M., Rogova, T., Shi, H., Sahara, N., Farley, A., Christensen, K., Duarte, F. and Dixon, D. J.
ChemRxiv, 2021, Preprint.

P2. Enantioselective synthesis of atropisomeric indoles via iron catalysed oxidative cross-coupling.
Surgenor, R., Liu, X., Myers, W. and Smith M. D.
ChemRxiv, 2021, Preprint.

P1. Intact nucleosomal context enables chromodomain reader MRG15 to distinguish H3K36me3 from -me2.
Faulkner, S., Couturier, A. M., Josephson, B., Watts, T., Davis, B. G. and Esashi, F.
bioRxiv, 2020, Preprint.

238. Photo-switchable anion binding and catalysis with a visible light responsive halogen bonding receptor.
Kerckhoffs, A., Moss, I. and Langton, M. J.
Chem. Commun., 2022, Accepted Manuscript.

237. Recent advances in the dearomative functionalisation of heteroarenes.
Kratena, N., Marinic, B. and Donohoe, T. J.
Chem. Sci., 2022, Advance Article.

236. Rapid and scalable halosulfonylation of strain-release reagents.
Pickford, H. D., Ripenko, V., McNamee, R. E., Holovchuk, S., Thompson, A. L., Smith, R. C., Mykhailiuk, P. K. and Anderson, E. A.
ChemRxiv, 2022, Preprint.
Angew. Chem. Int. Ed., 2022, Early View.

235. Rhodium-Catalyzed [2 + 2 + 2] Cyclotrimerizations of Yndiamides with Alkynes.
Smith, P. J., Tong, Z., Ragus, J., Solon, P., Shimkin, K. W. and Anderson, E. A.
Org. Lett., 2022, 24, 7522.

234. Enantioselective oxidation of unactivated C–H bonds in cyclic amines by iterative docking-guided mutagenesis of P450_BM3 (CYP102A1).
Zhang, Y., Xiong, Z., Li, Y., Wilson, M., Christensen, K. E., Jaques, E., Hernández-Lladó, P., Robertson, J. and Wong, L. L.
Nat. Synth., 2022, Accepted Article.

233. Fast relaxing red and near-IR switchable azobenzenes with chalcogen and halogen substituents: periodic trends, tuneable thermal half-lives and chalcogen bonding.
Kerckhoffs, A., Christensen, K. E. and Langton, M. J.
Chem. Sci., 2022, 13, 11551.

232. Synthesis of meta-substituted arene bioisosteres from [3.1.1]propellane.
Frank, N., Nugent, J., Shire, B.R., Pickford, H. D., Rabe, P., Sterling, A. J., Zarganes-Tzitzikas, T., Grimes, T., Thompson, A. L., Smith, R. C., Schofield, C. J., Brennan, P. E., Duarte, D. and Anderson, E. A.
ChemRxiv, 2022, Preprint.
Nature, 2022, 611, 721.

231. Identification of Histone Peptide Binding Specificity and Small-Molecule Ligands for the TRIM33α and TRIM33β Bromodomains.
Sekirnik, A., Reynolds, J., See, L., Bluck, J., Scorah, A., Tallant, C., Lee, B., Leszczynska, K., Grimley, R., Storer, R. I., Malattia, M, Crespillo, S., Caria, S., Duclos, S., Hammond, E. M., Knapp, S., Morris, G. M., Duarte, F., Biggin, P., and Conway, S. J.
ChemRxiv, 2022, Preprint.
ACS Chem. Biol., 2022, 17, 2753.

230. A One-Pot Synthesis-Functionalization Strategy for Streamlined Access to 2,5-Disubstituted 1,3,4-Oxadiazoles from Carboxylic Acids.
Matheau-Raven, D. and Dixon, D. J.
J. Org. Chem., 2022, 87, 12498.

229. Towards fully optimised and automated ESR spectroscopy.
Verstraete, J.-B., Yong, J. R. J., Goodwin, D. L., Myers, W. K. and Foroozandeh, M.
Chem. Commun., 2022, 58, 10715.

228. A Vicinal Diol Approach for the Total Synthesis of Molestin E, ent-Sinulacembranolide A and ent-Sinumaximol A.
Hoff, O., Kratena, N., Aynetdinova, D., Christensen, K. E. and Donohoe, T. J.
Chem. Eur. J., 2022, 28, e202202464.

227. Counterion-Mediated Enantioconvergent Synthesis of Axially Chiral Medium Rings.
Du, J.-Y., Balan, T., Claridge, T. D. W. C and Smith, M. D.
J. Am. Chem. Soc., 2022, 144, 14790.

226. N-Sulfinyl-O-(tert-Butyl)Hydroxylamine.
Davies, T. Q. and Willis, M. C.
In Encyclopedia of Reagents for Organic Synthesis. John Wiley & Sons, 2022.

225. An LNA-amide modification that enhances the cell uptake and activity of phosphorothioate exon-skipping oligonucleotides.
Baker, Y.R., Thorpe, C., Chen, J., Poller, L. M., Cox, L., Kumar, P., Lim, W. F., Lie, L., McClorey, G., Epple, S., Singleton, D., McDonough, M. A., Hardwick, J. S., Christensen, K. E., Wood, M. J. A., Hall, J. P., El-Sagheer, A. H., and Brown, T.
Nat. Commun., 2022, 13, 4036.

224. Alcohols as Alkylating Agents in the Cation-Induced Formation of Nitrogen Heterocycles.
Cox, L., Zhu, Y., Smith, P. J., Christensen, K. E., Sidera Portela, M. and Donohoe, T. J.
Angew. Chem. Int. Ed., 2022, 61, e202206800.

223. Branching out: redox strategies towards the synthesis of acyclic α-tertiary ethers.
Shennan, B. D. A., Berheci, D., Crompton, J. L., Davidson, T. A., Field, J. L., Williams, B. A and Dixon, D. J.
Chem. Soc. Rev., 2022, 51, 5878.

222. Modular Two-Step Route to Sulfondiimidamides.
Zhang, Z.-X., Bell, C., Ding, M. and Willis, M. C.
J. Am. Chem. Soc., 2022, 144, 11851.

221. An autonomously oscillating supramolecular self-replicator.
Howlett, M.G., Engwerda, A.H.J., Scanes, R.J.H. and Fletcher, S. P.
Nat. Chem., 2022, 14, 805.

220. Evolution of the Dearomative Functionalization of Activated Quinolines and Isoquinolines: Expansion of the Electrophile Scope.
Kischkewitz, M., Marinic, B., Kratena, N., Lai, Y., Hepburn, H. B., Dow, M., Christensen, K. E. and Donohoe,T. J.
Angew. Chem. Int. Ed., 2022, 61, e202204682.

219. Photocatalytic Late- Stage Functionalization of Sulfonamides via Sulfonyl Radical Intermediates.
Tilby, M.J ., Dewez, D. F., Pantaine, L. R. E., Hall, A., Martínez-Lamenca, C. and Willis, M. C.
ACS Catal., 2022, 12, 6060.

218. Extension of hydrogen borrowing alkylation reactions for the total synthesis of (−)-γ-lycorane.
Hall, C., Marriott, I., Christensen, K., Day, A., Goundry, W. and Donohoe, T. J.
Chem. Commun., 2022, 58, 4966.

217. [¹⁸F]Difluorocarbene for Positron Emission Tomography.
Sap, J.B.I., Meyer, C.F., Ford, J., Straathof, N., Dürr, A., Lelos, M., Paisey, S., Mollner, T., Hell, S., Trabanco, A., Genicot, C., am Ende, C., Paton, R. S., Tredwell, M. and Gouverneur, V..
Nature, 2022, 606, 102.

216. Transition Metal-Free, Visible Light-Mediated Radical Cyclisation of Malonyl Radicals onto 5-Ring Heteroaromatics.
Hernández-Lladó, P., Garrec, K., Schmitt, D. and Burton, J.
Adv. Synth. Catal., 2022, 364, 1724.

215. Reading and erasing of the phosphonium analogue of trimethyllysine by epigenetic proteins.
Kamps, J.J.A.G., Belle, R., Poater, J., Kumar, K., Pieters, B., Salah, E., Claridge, T. D. W., Paton, R., S., Bickelhaupt, F. M., Kawamura, A., Schofield, C. J. and Mecinović, J.
Commun. Chem., 2022, 5, 27.

214. Asymmetric Azidation under Hydrogen Bonding Phase-Transfer Catalysis: A Combined Experimental and Computational Study.
Wang, J., Horwitz, M. A., Dürr, A. B., Ibba, F., Pupo, G., Gao, Y., Ricci, P., Christensen, K. E., Pathak, T. P., Claridge, T. D. W. C., Lloyd-Jones, G. C., Paton, R. S. and Gouverneur, V.
J. Am. Chem. Soc., 2022, 144, 4572.

213. A Silyl Sulfinylamine Reagent Enables the Modular Synthesis of Sulfonimidamides via Primary Sulfinamides.
Ding, M., Zhang, Z.-X., Davies, T. Q. and Willis, M. C.
Org. Lett., 2022, 24, 1711.

212. Amino-oxetanes as amide isosteres by an alternative defluorosulfonylative coupling of sulfonyl fluorides.
Rojas, J. J., Croft, R. A., Sterling, A. J., Briggs, E. L., Antermite, D., Schmitt, D., Blagojevic, L., Haycock, P., White, A., Duarte, F., Choi, C., Mousseau, J. and Bull, J. A.
Nat. Chem., 2022, 14, 160.

211. DABSO – A Reagent to Revolutionize Organosulfur Chemistry.
Andrews, J. A. and Willis, M. C.
Synthesis, 2022, 54, 1695.

210. Modular Pulse Program Generation for NMR Supersequences.
Yong, J. R. J., Kupce, E. and Claridge, T. D. W.
Anal. Chem., 2022, 94, 2271.

209. Diverse saturated heterocycles from a hydroacylation/conjugate addition cascade.
Iwumene, N. U. N., Moseley, D. F., Pullin, R. C. and Willis, M. C.
Chem. Sci., 2022, 13, 1504.

208. Characterisation of the SARS-CoV-2 ExoN (nsp14^ExoN-nsp10) complex: implications for its role in viral genome stability and inhibitor identification.
Baddock, H., Brolih, S., Yosaatmadja, Y., Ratnaweera, M., Bielinski, M., Swift, L., Cruz-Migoni, A., Fan, H., Keown, J., Walker, A., Morris, G. M., Grimes, J., Fodor, E., Schofield, C. J., Gileadi, O. and McHugh, P. J.
bioRxiv, 2020, Preprint.
Nucleic Acids Res., 2022, 50, 1484.

207. A New Organocatalytic Desymmetrization Reaction Enables the Enantioselective Total Synthesis of Madangamine E.
Shiomi, S., Shennan, B., Yamazaki, K., Fuentes de Arriba, Á.L., Vasu, D., Hamlin, T. A. and Dixon, D. J.
ChemRxiv, 2021, Preprint.
J. Am. Chem. Soc., 2022, 144, 1407.

206. Bifunctional Iminophosphorane-Catalyzed Enantioselective Sulfa-Michael Addition to Unactivated α,β-Unsaturated Amides.
Rozsar, D., Formica, M., Yamazaki, K., Hamlin, T. and Dixon, D. J.
ChemRxiv, 2021, Preprint.
J. Am. Chem. Soc., 2022, 144, 1006.

205. Synthesis and Applications of Polysubstituted Bicyclo[1.1.0]butanes.
McNamee, R. E., Thompson, A. L. and Anderson E. A.
J. Am. Chem. Soc., 2021, 143, 21246.

204. Synthesis and Application of Constrained Amidoboronic Acids Using Amphoteric Boron-Containing Building Blocks.
Soor, H. S., Diaz, D. B., Tsui, K. Y., Calvopiña, K., Bielinski, M., Tantillo, D. J., Schofield, C. J. and Yudin, A. K.
J. Org. Chem., 2022, 87, 94.

203. Single photon double and triple ionization of allene.
Ideböhn, V., Sterling, A. J., Wallner, M., Olsson, E., Squibb, R. J., Miniotaite, U., Forsmalm, E., Forsmalm, M., Stranges, S., Dyke, J. M., Duarte, F., Eland, J. H. D., and Feifel, R.
Phys. Chem. Chem. Phys., 2022, 24, 786.

202. First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53.
Nowak, R., Tumber, A., Hendrix, E., Ansari, M., Sabatino, M., Antonini, L., Andrijes, R., Salah, E., Mautone, N., Pellegrini, F., Simelis, K., Kawamura, A., Johansson, C., Passeri, D., Pellicciari, R., Ciogli, A., Del Bufalo, D., Ragno, R., Coleman, M., Trisciuoglio, D., Mai, A., Oppermann, U., Schofield, C. J. and Rotili, D.
J. Med. Chem., 2021, 64, 17031.

201. Lactone Backbone Density in Rigid Electron-Deficient Semiconducting Polymers Enabling High n-type Organic Thermoelectric Performance.
Alsufyani, M., Stoeckel, M.-A., Chen, X., Thorley, K., Hallani, R.K., Puttisong, Y., Ji, X., Meli, D., Paulsen, B.D., Strzalka, J., Regeta, K., Combe, C., Chen, H., Tian, J., Rivnay, J., Fabiano, S. and McCulloch, I.
Angew. Chem. Int. Ed., 2022, 61, e202113078.

200. Parallel NMR Supersequences: Ten Spectra in a Single Measurement.
Kupče, E., Yong, J. R. J., Widmalm, G. and Claridge, T. D. W.
JACS Au, 2021, 1, 1892.

199. Electrophilic Activation of [1.1.1]Propellane for the Synthesis of Nitrogen-Substituted Bicyclo[1.1.1]pentanes.
Livesley, S., Sterling, A.J., Robertson, C.M., Goundry, W.R.F., Morris, J.A., Duarte, F. and Aïssa, C.
Angew. Chem. Int. Ed., 2022, 61, e202111291.

198. Benzenemethanamine, α,α-Diphenyl-N-Sulfinyl-.
Tilby, M. and Willis, M. C.
In Encyclopedia of Reagents for Organic Synthesis. John Wiley & Sons, 2021.

197. Synthesis of α-Quaternary Bicyclo[1.1.1]pentanes through Synergistic Organophotoredox and Hydrogen Atom Transfer Catalysis.
Nugent, J., Sterling, A. J., Frank, N., Mousseau, J. J. and Anderson, E. A.
Org. Lett., 2021, 23, 8628.

196. Sulfinates from Amines: A Radical Approach to Alkyl Sulfonyl Derivatives via Donor–Acceptor Activation of Pyridinium Salts.
Andrews, J., Pantaine, L., Palmer, C. F., Poole, D. L. and Willis, M. C.
Org. Lett., 2021, 23, 8488.

195. A Three-Component Ugi-Type Reaction of N-Carbamoyl Imines Enables a Broad Scope Primary α-Amino 1,3,4-Oxadiazole Synthesis.
Matheau-Raven, D., Boulter, E., Rogova, T. and Dixon, D. J.
Org. Lett., 2021, 23, 8209.

194. Red-shifted tetra-ortho-halo-azobenzenes for photo-regulated transmembrane anion transport.
Kerckhoffs, A., Bo, Z., Penty, S. E., Duarte, F. and Langton, M. J.
Org. Biomol. Chem., 2021, 19, 9058.

193. Exploiting Configurational Lability in Aza-Sulfur Compounds for the Organocatalytic Enantioselective Synthesis of Sulfonimidamides.
Tilby, M. J., Dewez, D. F., Hall, A., Martínez Lamenca, C. and Willis, M. C.
Angew. Chem. Int. Ed., 2021, 60, 25680.

192. A New 1,5-Disubstituted Triazole DNA Backbone Mimic with Enhanced Polymerase Compatibility.
Epple, S., Modi, A., Baker, Y. R., Wȩgrzyn, E., Traoré, D., Wanat, P., Tyburn, A., Shivalingam, A., Taemaitree, L., El-Sagheer, A. and Brown, T.
J. Am. Chem. Soc., 2021, 143, 16293.

191. Azine-N-oxides as effective controlling groups for Rh-catalysed intermolecular alkyne hydroacylation.
Moseley, D. F., Kalepua, J. and Willis, M. C.
Chem. Sci., 2021, 12, 13068.

190. Discovery of SARS-CoV-2 Mpro Peptide Inhibitors from Modelling Substrate and Ligand Binding.
Chan, H. T. H., Moesser, M., Walters, R. K., Malla, T. R., Twidale, R. M., John, T., Deeks, H. M., Johnston-Wood, T., Mikhailov, V., Sessions, R. B., Dawson, W., Salah, E., Lukacik, P., Strain-Damerell, C., Owen, D., Nakajima, T., Swiderek, K., Lodola, A., Moliner, V., Glowacki, D. R., Walsh, M. A., Schofield, C. J., Genovese, L., Shoemark, D., Mulholland, A. J., Duarte, F. and Morris, G. M.
bioRxiv, 2021, Preprint.
Chem. Sci., 2021, 12, 13686.

189. Regio- and stereoselective addition of Brønsted acids to yndiamides: Synthesis of N,O,N- and N,S,N-trisubstituted ketene acetals.
Garry, O. L., Mansfield, S. J. and Anderson, E. A.
Synthesis, 2021, 53, 4221.

188. Switchable, Reagent-Controlled Diastereodivergent Photocatalytic Carbocyclisation of Imine-Derived α-Amino Radicals.
Maitland, J. A. P., Leitch, J. A., Yamazaki, K., Christensen, K. E., Cassar, D. J., Hamlin, T. A. and Dixon, D. J.
Angew. Chem. Int. Ed., 2021, 60, 24116.

187. X-ray free-electron laser studies reveal correlated motion during isopenicillin N synthase catalysis.
Rabe, P., Kamps, J. J. A. G., Sutherlin, K., Linyard, J., Aller, P., Pham, C., Makita, H., Clifton, I., McDonough, M., Leissing, T., Shutin, D., Lang, P., Butryn, A., Brem, J., Gul, S., Fuller, F., Kim, I-S., Cheah, M., Fransson, T., Bhowmick, A., Young, I., O’Riordan, L., Brewster, A., Pettinati, I., Doyle, M., Joti, Y., Owada, S., Tono, K., Batyuk, A., Hunter, M., Alonso-Mori, r., Bergmann, U., Owen, R., Sauter, N., Claridge, T. D. W., Robinson, C. V., Yachandra, V. K., Yano, J., Kern, J. F., Orville, A. M. and Schofield, C. J.
Sci. Adv., 2021, 7, eabh0250.

186. Selection between Competing Self-Reproducing Lipids: Succession and Dynamic Activation.
Howlett, M. G., Scanes, R. J. H. and Fletcher, S. P.
JACS Au, 2021, 1, 1355.

185. A phosphate binding pocket is a key determinant of exo- versus endo-nucleolytic activity in the SNM1 nuclease family.
Baddock, H., Newman, J., Yosaatmadja, Y., Bielinski, M., Schofield, C. J., Gileadi, O and McHugh, P. J.
Nucleic Acids Res., 2021, 49, 9294.

184. Structural and mechanistic insights into the Artemis endonuclease and strategies for its inhibition.
Yosaatmadja, Y., Baddock, H., Newman, J., Bielinski, M., Gavard, A., Mukhopadhyay, S., Dannerfjord, A., Schofield, C. J., McHugh, P. J. and Gileadi, O.
bioRxiv, 2021, Preprint.
Nucleic Acids Res., 2021, 49, 9310.

183. Synthesis of Polysubstituted Fused Pyrroles by Gold-Catalyzed Cycloisomerization/1,2-Sulfonyl Migration of Yndiamides.
Smith, P. J., Jiang, Y., Tong, Z., Pickford, H. D., Christensen, K. E., Nugent, J. and Anderson, E. A.
Org. Lett., 2021, 23, 6547.

182. Base-Activated Latent Heteroaromatic Sulfinates as Nucleophilic Coupling Partners in Palladium-Catalyzed Cross-Coupling Reactions.
Cook, X. A. F., Pantaine, L. R. E., Blakemore, D. C., Moses, I. B., Sach, N. W., Shavnya, A. and Willis, M. C.
Angew. Chem. Int. Ed., 2021, 60, 22461.

181. On-the-Fly, Sample-Tailored Optimization of NMR Experiments.
Yong, J. R. J. and Foroozandeh, M.
Anal. Chem., 2021, 93, 10735.

180. Supramolecular chemistry in lipid bilayer membranes.
Kerckhoffs, A., Bickerton, L., Johnson, T. and Langton, M. J.
Chem. Sci., 2021, 12, 11252.

179. Artificial nucleic acid backbones and their applications in therapeutics, synthetic biology and biotechnology.
Epple, S., El-Sagheer, A. H. and Brown, T.
Emerg. Top. Life Sci., 2021, 5, 691.

178. An on-demand, drop-on-drop method for studying enzyme catalysis by serial crystallography.
Butryn, A., Simon, P., Aller, P., Hinchliffe, P., Massad, R., Leen, G., Tooke, C., Bogacz, I., Kim, I-S., Bhowmick, A., Brewster, A. S., Devenish, N., Brem, J., Kamps, J., Lang, P., Rabe, P., Axford, D., Beale, J., Davy, B., Ebrahim, A., Orlans, J., Storm, S., Zhou, T., Owada, S., Tanaka, R., Tono, K., Evans, G., Owen, R., Houle, F., Sauter, N., Schofield, C. J., Spencer, J., Yachandra, V., Yano, J., Kern, J. and Orville, A. M.
Nat. Commun., 2021, 12, 4461.

177. A General Iridium-Catalyzed Reductive Dienamine Synthesis Allows a Five-Step Synthesis of Catharanthine via the Elusive Dehydrosecodine.
Gabriel. P., Almehmadi, Y., Rong Wong, Z. and Dixon, D. J.
J. Am. Chem. Soc., 2021, 143, 10828.

176. Controlling Intramolecular Interactions in the Design of Selective, High-Affinity, Ligands for the CREBBP Bromodomain.
Brand, M., Clayton, J., Moroglu, M., Schiedel, M., Picaud, S., Bluck, J., Skwarska, A., Bolland, H., Chan, A., Laurin, C., Scorah, A., See, L., Rooney, T., Andrews, K., Fedorov, O., Perell, G., Kalra, P., Vinh, K., Cortopassi, W., Heitel, P., Christensen, K., Cooper, R., Paton, R., Pomerantz, W., Biggin, P., Hammond, E. M., Filippakopoulos, P. and Conway, S. J.
ChemRxiv, 2020, Preprint.
J. Med. Chem., 2021, 64, 10102.

175. How do we address neglected sulfur pharmacophores in drug discovery?
Tilby, M. J. and Willis, M. C.
Expert Opin. Drug Discov., 2021, 16, 1227.

174. A catalytic asymmetric cross-coupling approach to the synthesis of cyclobutanes.
Goetzke, F.W., Hell, A.M.L., van Dijk, L. and Fletcher, S. P.
Nat. Chem., 2021, 13, 880.

173. General α-Amino 1,3,4-Oxadiazole Synthesis via Late-Stage Reductive Functionalization of Tertiary Amides and Lactams.
Mattheau-Raven, D. and Dixon, D. J.
ChemRxiv, 2021, Preprint.
Angew. Chem. Int. Ed., 2021, 60, 19725.

172. Twofold Radical-Based Synthesis of N,C-Difunctionalized Bicyclo[1.1.1]pentanes.
Pickford, H. D., Nugent, J., Owen, B., Mousseau, J. J., Smith, R. C. and Anderson, E. A.
J. Am. Chem. Soc., 2021, 143, 9729.

171. Increasing Sensitivity and Versatility in NMR Supersequences with New HSQC-based Modules.
Yong, J. R. J., Hansen, A. L., Kupče, E. and Claridge, T. D. W. C.
J. Magn. Reson., 2021, 329, 107027.

170. Rh-catalyzed asymmetric Suzuki-Miyaura cross-coupling.
Van Dijk, L. and Fletcher, S. P.
Trends Chem., 2021, 3, 795.

169. General Pyrrolidine Synthesis via Iridium-Catalyzed Reductive Azomethine Ylide Generation from Tertiary Amides and Lactams.
Gabriel, P., Yamazaki, K., Di Carmine, G., Pedroni, J., Farizyan, M., Hamlin, T. and Dixon, D. J.
ChemRxiv, 2021, Preprint.
ACS Catal., 2021, 11, 7489.

168. Au(I)-Catalyzed Oxidative Functionalization of Yndiamides.
Tong, Z., Garry, O., Smith, P. J., Jiang, Y, Mansfield, S. J. and Anderson, E. A.
Org. Lett., 2021, 23, 4888.

167. Late-stage difluoromethylation: concepts, developments and perspective.
Sap, J., Meyer, C., Straathof, N., Iwumene, N., am Ende, C., Trabanco, A. and Gouverneur, V.
Chem. Soc. Rev., 2021, 50, 8214.

166. Highly Active Halogen Bonding and Chalcogen Bonding Chloride Transporters with Non-Protonophoric Activity.
Bickerton, L., Docker, A., Sterling, A. J., Kuhn, H., Duarte, F., Beer, P. D. and Langton, M. J.
Chem. Eur. J., 2021, 27, 11738.

165. Acceleration of lipid reproduction by emergence of microscopic motion.
Babu, D., Scanes, R.J.H., Plamont, R., Ryabchun, A., Lancia, F., Kudernac, T., Fletcher, S.P. and Katsonis, N.
Nat. Commun., 2021, 12, 2959.

164. Synthesis of 1,3-disubstituted bicyclo[1.1.0]butanes via directed bridgehead functionalization.
McNamee, R. E., Haugland, M. M., Nugent, J., Chan, R., Christensen, K. E. and Anderson, E. A.
Chem. Sci., 2021, 12, 7480.

163. Rediscovering Sulfinylamines as Reagents for Organic Synthesis.
Davies, T. Q. and Willis, M. C.
Chem. Eur. J., 2021, 27, 8918.

162. A Novel Automated Screening Method For Combinatorial Small Molecules.
Yu, P., Sterling, A. and Hein, J.
ChemRxiv, 2020, Preprint.
J. Chem. Inf. Model., 2021, 61, 1637.

161. Parallel nuclear magnetic resonance spectroscopy.
Kupče, Ē., Frydman, L., Webb, A.G., Yong, J.R.J. and Claridge, T.D.W.
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160. Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications.
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159. Mechanistic investigation of Rh(I)-catalysed asymmetric Suzuki–Miyaura coupling with racemic allyl halides.
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158. Chemogenomics for drug discovery: clinical molecules from open access chemical probes.
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157. A Bifunctional Iminophosphorane Squaramide Catalyzed Enantioselective Synthesis of Hydroquinazolines via Intramolecular Aza-Michael Addition to α,β-Unsaturated Esters.
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156. Direct catalytic asymmetric synthesis of α-chiral bicyclo[1.1.1]pentanes.
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155. Installing the “magic methyl” – C–H methylation in synthesis.
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154. Hydrogen borrowing catalysis using 1° and 2° alcohols: Investigation and scope leading to α and β branched products.
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153. Selectivity in organocatalysis - From qualitative to quantitative predictive models.
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152. Hydrogen Borrowing Alkylation of 1,2‐Amino Alcohols in the Synthesis of Enantioenriched γ‐Aminobutyric Acids.
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151. Synthesis of legonmycins A and B, C(7a)-hydroxylated bacterial pyrrolizidines.
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150. Mass spectrometry reveals potential of β-lactams as SARS-CoV-2 M^pro inhibitors.
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149. Masked Alkyne Equivalents for the Synthesis of Mechanically Interlocked Polyynes.
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148. Advances in polycyclization cascades in natural product synthesis.
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147. Single point activation of pyridines enables reductive hydroxymethylation.
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146. autodE: Automated Calculation of Reaction Energy Profiles – Application to Organic and Organometallic Reactions.
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145. Cyclic Peptides as Chemical Probes.
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144. Primary Sulfonamide Synthesis Using the Sulfinylamine Reagent N-Sulfinyl-O-(tert-butyl)hydroxylamine, t-BuONSO.
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143. Fragment-Based Identification of Ligands for Bromodomain-Containing Factor 3 of Trypanosoma Cruzi.
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142. A Single‐Stranded DNA‐Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks.
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141. Synthesis and Structure–Activity Relationship of Dehydrodieugenol B Neolignans against Trypanosoma cruzi.
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140. Enzymatic Kinetic Resolution by Addition of Oxygen.
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139. Inhibition of the SUV4-20 H1 histone methyltransferase increases frataxin expression in Friedreich’s ataxia patient cells.
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138. The 2‐Pyridyl Problem: Challenging Nucleophiles in Cross‐Coupling Arylations.
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137. α-Tertiary Dialkyl Ether Synthesis via Reductive Photocatalytic α-Functionalization of Alkyl Enol Ethers.
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136. Bifunctional Iminophosphorane Superbase Catalysis: Applications in Organic Synthesis.
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135. Visible light mediated heterocycle functionalization via a geometrically interrupted [2+2] cycloaddition.
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134. Reverse Polarity Reductive Functionalization of Tertiary Amides via a Dual Iridium-Catalyzed Hydrosilylation and Single Electron Transfer Strategy.
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133. Harnessing Sulfinyl Nitrenes: A Unified One-Pot Synthesis of Sulfoximines and Sulfonimidamides.
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132. Super-resolution RESOLFT microscopy of lipid bilayers using a fluorophore-switch dyad.
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131. Rhodium catalysed C-3/5 methylation of pyridines using temporary dearomatisation.
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130. A Modular and Divergent Approach to Spirocyclic Pyrrolidines.
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129. Synthesis of Fluorinated Alkyl Aryl Ethers by Palladium-Catalyzed C–O Cross-Coupling.
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128. Catalytic Reductive Functionalization of Tertiary Amides using Vaska’s Complex: Synthesis of Complex Tertiary Amine Building Blocks and Natural Products.
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127. Coupled metabolic cycles allow out‐of‐equilibrium autopoietic vesicle replication.
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126. Selective fragments for the CREBBP bromodomain identified from an Encoded Self‑Assembly Chemical Library.
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125. A Heck reaction/photochemical alkene isomerization sequence to prepare functionalized quinolines.
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124. Controlling gene expression with light: a multidisciplinary endeavour.
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123. Synthesis of Cyclo[18]carbon via Debromination of C₁₈Br₆.
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122. Atropisomerism in diarylamines: structural requirements and mechanisms of conformational interconversion.
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121. Hydrogen Bonding Phase-Transfer Catalysis with Ionic Reactants: Enantioselective Synthesis of γ-Fluoroamines.
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120. Single‐molecule observation of intermediates in bioorthogonal 2‐cyanobenzothiazole chemistry.
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119. BIMP Catalyzed 1,3-Prototropic Shift for the Highly Enantioselective Synthesis of Conjugated Cyclohexenones.
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118. Structure-activity relationship study of cytotoxic neolignan derivatives using multivariate analysis and computation-aided drug design.
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117. Reversible photo-control over transmembrane anion transport using visible-light responsive supramolecular carriers.
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116. Engineered anti-inflammatory peptides inspired by mapping an evasin-chemokine interaction.
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115. α‐Amidoaldehydes as substrates in rhodium‐catalyzed intermolecular alkyne hydroacylation: The synthesis of α‐amidoketones.
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114. Palladium-Catalyzed Desulfinative Cross-Couplings.
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113. Organophotochemical S_NAr Reactions of Mildly Electron‐Poor Fluoroarenes.
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112. Synthesis of All-carbon Disubstituted Bicyclo[1.1.1]pentanes by Iron-Catalyzed Kumada Cross-Coupling.
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111. Control of Absolute Stereochemistry in Transition‐Metal‐Catalyzed Hydrogen Borrowing Reactions.
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110. Consecutive 5′- and 3′-amide linkages stabilise antisense oligonucleotides and elicit an efficient RNase H response.
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109. Transmembrane anion transport mediated by halogen bonding and hydrogen bonding triazole anionophores.
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108. Rationalizing the diverse reactivity of [1.1.1]propellane through sigma-pi-delocalization.
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107. Enantiomerically Enriched Tetrahydropyridine Allyl Chlorides.
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106. An Asymmetric Suzuki–Miyaura Approach to Prostaglandins: Synthesis of Tafluprost.
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105. A hydrogen borrowing annulation strategy for the stereocontrolled synthesis of saturated aza-heterocycles.
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104. Enantioconvergent alkylation of ketones with racemic secondary alcohols via hydrogen borrowing catalysis.
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103. Double and triple ionization of isocyanic acid.
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102. Mechanistic Studies of the Palladium-Catalyzed Desulfinative Cross-Coupling of Aryl Bromides and (Hetero)Aryl Sulfinate Salts.
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101. A Modular, Enantioselective Synthesis of Resolvins D3, E1, and Hybrids.
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100. Synthesis of the cyclopentane core of pepluanin A.
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99. Chemo- and Regioselective Synthesis of Acyl-Cyclohexenes by a Tandem Acceptorless Dehydrogenation-[1,5]-Hydride Shift Cascade.
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98. [1.1.1]Propellane.
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97. α-Amino Radicals via Photocatalytic Single-Electron Reduction of Imine Derivatives.
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96. Bicyclic Lactams Derived from Serine or Cysteine and 2-Methylpropanal.
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95. Inhibitors of JmjC-Containing Histone Demethylases.
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94. ¹⁸F-Trifluoromethanesulfinate Enables Direct C–H ¹⁸F-Trifluoromethylation of Native Aromatic Residues in Peptides.
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93. Dearomative Photocatalytic Construction of Bridged 1,3-Diazepanes.
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92. Catalytic Asymmetric Suzuki–Miyaura Couplings.
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91. Structural Insights into Interaction Mechanisms of Alternative Piperazine-urea YEATS Domain Binders in MLLT1.
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90. Iridium-Catalyzed Reductive Coupling of Grignard Reagents and Tertiary Amides.
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89. Synthesis of highly fluorinated arene complexes of [Rh(chelating phosphine)]+ cations, and their use in synthesis and catalysis.
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88. ¹⁹F NMR studies on γ-butyrobetaine hydroxylase provide mechanistic insights and suggest a dual inhibition mode.
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87. How formaldehyde reacts with amino acids.
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86. Characterisation of utrophin modulator SMT C1100 as a non-competitive inhibitor of firefly luciferase.
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85. Synthesis of Cyclic Alkenyl Dimethylsiloxanes from Alkynyl Benzyldimethylsilanes and Application in Polyene Synthesis
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84. Convergent Total Syntheses of (−)‐Rubriflordilactone B and (−)‐pseudo‐Rubriflordilactone B
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83. Highly enantioselective rhodium-catalyzed cross-coupling of boronic acids and racemic allyl halides.
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82. A General Route to Bicyclo[1.1.1]pentanes through Photoredox Catalysis
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81. Desymmetrization of Meso-bisphosphates via Rhodium Catalyzed Asymmetric Allylic Arylation
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80. Bicyclic Boronate VNRX-5133 Inhibits Metallo- and Serine-β-Lactamases
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79. Modular Sulfondiimine Synthesis Using a Stable Sulfinylamine Reagent
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78. Iridium-Catalyzed Aza-Spirocyclization of Indole-Tethered Amides: An Interrupted Pictet–Spengler Reaction
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77. Retooling Asymmetric Conjugate Additions for Sterically Demanding Substrates with an Iterative Data-Driven Approach
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76. Rhodium-catalysed vinyl 1,4-conjugate addition coupled with Sharpless asymmetric dihydroxylation in the synthesis of the CDE ring fragment of pectenotoxin-4
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75. Synthesis and biophysical properties of carbamate-locked nucleic acid (LNA) oligonucleotides with potential antisense applications
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74. Intramolecular Aldol Ring Closures of Cysteine Derivatives Leading to Densely Functionalised Pyroglutamates
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73. Total Synthesis of Berkeleylactone A
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72. Dehydrodieugenol B derivatives as antiparasitic agents: Synthesis and biological activity against Trypanosoma cruzi
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71. A General Copper-Catalyzed Synthesis of Ynamides from 1,2-Dichloroenamides​
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70. A halogen-bonding foldamer molecular film for selective reagentless anion sensing in water
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69. Synthesis of Enantioenriched α‐Chiral Bicyclo[1.1.1]pentane​​
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68. A chemically fuelled self-replicator
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67. Practical and scalable kinetic resolution of BINOLs mediated by a chiral counterion
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66. Dithiane-Directed Rh(III)-Catalyzed Amidation of Unactivated C(sp3)-H Bonds
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Chem. Sci., 2019, 10, 3733.

65. The fluorination of C–H bonds: developments and perspectives​
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64. Primary α-Tertiary Amine Synthesis via α-C–H Functionalization
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63. Anion recognition in water by charge-neutral halogen and chalcogen bonding foldamer receptors​
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62. Chemical Probes​
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61. Hydrogen Bonding Phase-Transfer Catalysis with Potassium Fluoride: Enantioselective Synthesis of β-Fluoroamines
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60. Conformational Effects on Physical-Organic Descriptors – the Case of Sterimol Steric Parameters​
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59. Hydrogen bond enabled dynamic kinetic resolution of axially chiral amides mediated by a chiral counterion
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Angew. Chem. Int. Ed., 2019, 58, 2795.

58. Chemical epigenetics: the impact of chemical‐ and chemical biology techniques on bromodomain target validation​
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57. Desymmetrization of meso-bisphosphates using copper catalysis and alkylzirconocene nucleophiles
Jacques, R., Pullin, R. D. C. and Fletcher, S. P.
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56. Data-mining the diaryl(thio)urea conformational landscape: Understanding the contrasting behavior of ureas and thioureas with quantum chemistry
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Tetrahedron, 2019, 75, 697.

55. Non‐Hydrolytic β‐Lactam Antibiotic Fragmentation by L,D‐Transpeptidases and Serine β‐Lactamase Cysteine Variants
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54. Enantioselective rhodium-catalysed insertion of trifluorodiazoethanes into tin hydrides
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Tetrahedron, 2019, 75, 17.

53. Design, Synthesis and Characterization of Covalent KDM5 Inhibitors
Wright, M., Vazquez-Rodriguez, S., Rogers, C. M., Cribbs, A., Velupillai, S., Philpott, M., Lee, H., Dunford, J. E., Huber, K. V. M., Robers, M. B., Vasta, J. D., Thezenas, M.-L., Bonham, S., Kessler, B., Bennett, J., Fedorov, O., Raynaud, F., Donovan, A., Blagg, J., Bavetsias, V., Oppermann, U., Kawamura, A. and Brennan, P. E.
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52. A structure-based approach towards identification of inhibitory fragments for eleven-nineteen-leukemia protein (ENL)
Heidenreich, H., Moustakim, M., Schmidt, J., Merk, D., Brennan, P. E., Fedorov, O., Chaikuad, A. and Knapp, S.
J. Med. Chem., 2018, 61, 10929.

51. Target Identification Using Chemical Probes​
Moustakim, M., Ling Felce, S., Zaarour, N., Farnie, G., McCann, F. E. and Brennan, P. E.
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50. Stereospecific 1,3-H Transfer of Indenols Proceeds via Persistent Ion-Pairs Anchored By NH···Pi Interactions
Ascough, D. M. H., Duarte, F. and Paton, R. S.
ChemRxiv, 2018, Preprint.
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49. Copper-catalysed synthesis of alkylidene 2-pyrrolinone derivatives from the combination of α-keto amides and alkynes
Tan, Q. W., Chovatia, P. and Willis, M. C.
Org. Biomol. Chem., 2018, 16, 7797.

48. Discovery of an MLLT1/3 YEATS Domain Chemical Probe
Moustakim, M., Christott, T., Monteiro, O. P., Bennett, J., Giroud, C., Ward, J., Rogers, C. M., Smith, P., Panagakou, I., Saez, L. D., Ling Felce, S., Gamble, V., Gileadi, C., Halidi, N., Heidenreich, D., Chaikuad, A., Knapp, S., Huber, K. V. M., Farnie, G., Heer, J., Manevski, N., Poda, G., Al-awar, R., Dixon, D. J., Brennan, P. E. and Fedorov, F.
ChemRxiv, 2018, Preprint.
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47. Enantioselective Silver-Catalyzed Cascade Synthesis of Fused Lactone and Lactam Oxazolines
de la Campa, R., Manzano, R., Calleja, P., Ellis, S. R. and Dixon, D. J.
Org.Lett., 2018, 20, 6033.

46. Post-translational site-selective protein backbone α-deuteration
Galan, S. R. G., Wickens, J. R., Dadova, J., Ng, W.-L., Zhang, X., Simion, R. A., Quinlan, R., Pires, E., Paton, R. S., Caddick, S., Chudasama, V. and Davis. B. G.
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45. Principles and Applications of Fragment-based Drug Discovery for Chemical Probes
Moustakim, M. and Brennan, P. E.
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44. Bifunctional Iminophosphorane Catalysed Enantioselective Sulfa-Michael Addition of Alkyl Thiols to Alkenyl Benzimidazoles
Formica, M., Sorin, G., Farley, A. J. M., Díaz, J., Paton, R. S. and Dixon, D. J.
Chem. Sci., 2018, 9, 6969.

43. Photocatalytic Reverse Polarity Povarov Reaction
Leitch, J. A., Fuentes de Arriba, A. L., Tan, J., Hoff, O., Martínez, C. M. and Dixon, D. J.
Chem. Sci., 2018, 9, 6653.

42. Polyyne formation via skeletal rearrangement induced by atomic manipulation
Pavliček, N., Gawel, N., Kohn, D. R., Majzik, Z., Xiong, Y., Meyer, G., Anderson, H. L. and Gross, L.
Nat. Chem., 2018, 10, 853.

41. A Bench-Stable Transfer Reagent for the Synthesis of Trifluoromethyl-sulfonimidamides from Sulfinamides
Wright, M., Martinez-Lamenca, C., Leenaerts, J. E., Brennan, P. E., Trabanco, A. A., Oehlrich, D.
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40. A transient self-assembling self-replicator
Colomer, I., Morrow, S. M. and Fletcher S. P.
Nat. Commun., 2018, 9, 2239.

39. The Plant Cysteine Oxidases from Arabidopsis thaliana are kinetically tailored to act as oxygen sensors
White, Mark. D., Kamps, J. A. G., East, S., Taylor Kearney, L. J. and Flashman, E.
J. Biol. Chem., 2018, 293, 11786.

38. Roles of 2-oxoglutarate oxygenases and isopenicillin N synthase in β-lactam biosynthesis
Rabe, P., Kamps, J. A. G., Schofield, C. J. and Lohans, C. T.
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37. Synthesis and Applications of Highly Functionalized 1-Halo-3-Substituted Bicyclo[1.1.1]pentanes
Caputo, D. F. J., Arroniz, C., Dürr, A. B., Mousseau, J. J., Stepan, A. F., Mansfield, S. J. and Anderson, E. A.
Chem. Sci., 2018, 9, 5295.

36. Rh(DPEPhos)-Catalyzed Alkyne Hydroacylation using β-Carbonyl Substituted Aldehydes. Mechanistic Insight Leads to Low Catalyst Loadings that Enables Selective Catalysis on Gram-Scale
Barwick-Silk, J., Hardy, S., Willis, M. C. and Weller, A., S.
J. Am. Chem. Soc., 2018, 140, 7347

35. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
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34. Asymmetric nucleophilic fluorination under hydrogen bonding phase-transfer catalysis
Ascough, D. M. H., Pupo, G., Ibba, F., Vicini, A. C., Ricci, P., Christensen, K. E., Pfeifer, L. Morphy, J. R., Brown, J. M., Paton, R. S. and Gouverneur, V.
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33. An enamine controlling group for rhodium-catalyzed intermolecular hydroacylation
Straker, R. N., Formica, M., Lupton, J. D., Niu, J. and Willis, M. C.
Tetrahedron, 2018, 74, 5408.

32. Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2
Moustakim, M., Riedel, K., Schuller, M., Gehring, A. P., Monteiro, O. P., Martin, S. P., Fedorov, O., Heer, J., Dixon, D. J., Elkins, J. M., Knapp, S., Bracher, F. and Brennan, P. E.
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31. Molecular machines for catalysis
van Dijk, L., Tilby, M. J., Szpera, R., Smith, O. A., Bunce, H. A. P. and Fletcher, S. P.
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30. Structure activity relationship studies on rhodanines and derived enethiol inhibitors of metallo-β-lactamases
Zhang, D., Markoulides, M. S., Stepanovs, D., Rydzik, A. M., El-Hussein, A., Bon, C., Kamps, J. J. A. G., Umland, K.-D., Collins, P. M., Cahill, S. T., Wanga, D. Y., von Delft, F., Brem, J., McDonough, M. A. and Schofield, C. J.
Bioorg. Med. Chem., 2018, 26, 2928.

29. Spironaphthoxazine switchable dyes for biological imaging
Xiong, Y., Vargas Jentzsch, A., Osterrieth, J. W. M., Sezgin, E., Sazanovich, I. W., Reglinski, K., Galiani, S., Parker, A. W., Eggeling, C. and Anderson, H. L.
Chem. Sci., 2018, 9, 3029.

28. Formation of quaternary centres by copper catalysed asymmetric conjugate addition to β-substituted cyclopentenones with the aid of a quantitative structure–selectivity relationship
Ardkhean, R., Mortimore, M., Paton, R. S. and Fletcher, S. P.
Chem. Sci., 2018, 9, 2628.

27. Synthesis of Polyynes Using Dicobalt Masking Groups
Kohn, D. R., Gawel, P., Xiong, Y., Christensen, K. E. and Anderson, H. L.
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26. Detecting Mechanochemical Atropisomerization within an STM Break Junction
Leary, E., Roche, C., Jiang, H., Grace, I., González, M. T., Rubio-Bollinger, G., Romero-Muñiz, C., Xiong, Y., Al-Galiby, Q., Noori, M., Lebedeva, M. A., Porfyrakis, K., Agrait, N., Hodgson, A., Higgins, S. J., Lambert, C. J., Anderson, H. L. and Nichols, R. J
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25. Total synthesis of (−)-himalensine A
Shi, H., Michaelides, I. N., Darses, B., Jakubec, P., Nguyen, Q. N. N., Paton, R. S. and Dixon, D. J.
J. Am. Chem. Soc. 2017, 139, 17755.

24. Hexafluoroisopropanol as a highly versatile solvent
Colomer, I., Chamberlain, A. E. R., Haughey, M. B., Donohoe, T. J.
Nature Rev. Chem. 2017, 1, 0088.

23. One-pot, Three-Component Sulfonimidamide Synthesis exploiting the Sulfinylamine Reagent N-Sulfinyltritylamine, TrNSO
Davies, T. Q., Hall, A. and Willis, M. C.
Angew. Chem. Int. Ed. 2017, 56, 14937.

22. Copper-Catalyzed Synthesis and Applications of Yndiamide
Mansfield, S. J., Christensen, K. E., Thompson, A. L., Ma, K., Jones, M. W., Mekareeya, A. and Anderson​, E. A.
Angew. Chem. Int. Ed. 2017, 56, 14428.

21. Enantioselective Conjugate Addition Catalyzed by a Copper Phosphoramidite Complex: Computational and Experimental Exploration of Asymmetric Induction
Ardkhean, R.,  Roth, P. M. C., Maksymowicz, R. M., Curran, A., Peng, Q., Paton, R. S. and Fletcher, S. P.
ACS Catal. 2017, 7, 6729.

20. Crotonases - Nature's Exceedingly Convertible Catalysts
Lohans, C. T., Wang, D. Y., Wang, J., Hamed, R. B., Schofield, C. J.
ACS Catal. 2017, 7, 6587.

19. Exploiting Carbonyl Groups to Control Intermolecular Rhodium-Catalyzed Alkene and Alkyne Hydroacylation
Coxon, T. J., Fernandez, M., Barwick-Silk, J., McKay, A. I., Britton, L. E., Weller, A. S., Willis, M. C.
J. Am. Chem. Soc. 2017, 139, 10142.

18. Visible light photocatalysis of 6π heterocyclization
Münster, N., Parker, N. A., van Dijk, L., Paton, R. S., Smith, M. D.
Angew. Chem. Int. Ed. 2017, 56, 9468.

17. Unexpected Interactions between Alkyl Straps and Pyridine Ligands in Sulfur-Strapped Porphyrin Nanorings
Roche, C., Lou, Q., Gil-Ramirez, G., Jiang, H.-W., Kohn, D. R., Xiong, Y., Thompson, A. L., Anderson, H. L.
J. Org. Chem. 2017, 82, 7446.

16. Potential for minimal self-replicating systems in a dynamic combinatorial library of equilibrating imines
Morrow, S. M., Bissette, A. J., Fletcher, S. P.
Tetrahedron 2017, 73, 5005.

15. Transmission of chirality through space and across length scales
Morrow, S. M., Bissette, A. J. and Fletcher, S. P.
Nature Nanotechnology 2017, 12, 410.

14. Structural and stereoelectronic insights into oxygenase-catalyzed formation of ethylene from 2-oxoglutarate
Zhang, Z., Smart, T. J., Choi, H., Hardy, F., Lohansa, C. T., Abboud, M. I., Richardson, M. S. W., Paton, R. S., McDonough, M. A. and Schofield, C. J.
Proc. Natl. Acad. Sci. 2017, 114, 4667. 

13. Neutral iodotriazole foldamers as tetradentate halogen bonding anion receptors
Borissov, A., Lim, J. Y. C., Brown, A., Christensen, K. E., Thompson, A. L., Smith, M. D. and Beer, P. D.
Chem. Commun. 2017, 53, 2483.

12. Discovery of a PCAF Bromodomain Chemical Probe
Moustakim, M., Clark, P. G. K., Trulli, L., Fuentes de Arriba, A. L., Ehebauer, M. T., Chaikuad, A., Murphy, E. J., Mendez-Johnson, J., Daniels, D., Hou, C.-F. D., Lin, Y.-H., Walker, J. R., Hui, R., Yang, H., Dorrel, L., Rogers, C. M., Monteiro, O. P., Fedorov, O., Huber, K. V. M., Knapp, S., Heer, J., Dixon, D. J., Brennan, P. E.
Angew. Chem. Int. Ed. 2017, 56, 827. DOI: 10.1002/anie.201610816.

11. Umpolung synthesis of branched α-functionalized amines from imines via photocatalytic three-component reductive coupling reactions
Fuentes de Arriba, A. L., Urbitsch, F., Dixon, D. J.
Chem. Commun. 2016, 52, 14434.

10. A Cascade Strategy Enables a Total Synthesis of (+/-)-Morphine
Chu, S., Münster, N., Balan, T., Smith. M. D.
Angew. Chem. Int. Ed. 2016, 55, 14306.

9. Posttranslational mutagenesis: A chemical strategy for exploring protein side-chain diversity
Wright, T. H., Bower, B. J., Chalker, J. M., Bernardes, G. J. L., Wiewiora, R., Ng, W.-L., Raj, R., Faulkner, S., Vallée, M. R. J., Phanumartwiwath, A., Coleman, O. D., Thézénas, M.-L., Khan, M., Galan, S. R. G., Lercher, L., Schombs, M. W., Gerstberger, S., Palm-Espling, M. E., Baldwin, A. J., Kessler, B. M., Claridge, T. D. W., Mohammed, S. and Davis, B. G.
Science 2016, 354, 597.

8. Chemical Probes and Inhibitors of Bromodomains outside the BET family
Moustakim, M., Clark, P. G. K., Hay, D. A., Dixon, D. J. and Brennan, P. E.
Med. Chem. Commun. 2016, 7, 2246.

7. Photoswitchable Spiropyran Dyads for Biological Imaging
Xiong, Y., Rivera-Fuentes, P., Sezgin, E., Jentzsch, A. V., Eggeling, C. and Anderson, H. L.
Org. Lett. 2016, 8, 3666.

6. Cp₂ZrMeCl: A Reagent for Asymmetric Methyl Addition
Garrec, K. and Fletcher, S. P.
Org. Lett. 2016, 8, 3814.

5. Recent Applications in Natural Product Synthesis of Dihydrofuran and -pyran Formation by Ring-closing Alkene Metathesis
Jacques, R., Pal, R., Parker, N. A., Sear, C. E., Smith, P. W., Ribaucourt, A. and Hodgson, D. M.
Org. Biomol. Chem. 2016, 14, 5875.

4. Organocatalytic Enantioselective Desymmetrisation
Borissov, A., Davies, T. Q., Ellis, S. R., Fleming T. F., Richardson, M. S. W. and Dixon, D. J.
Chem. Soc. Rev. 2016, 45, 5474.

3. Cascade Polycyclizations in Natural Product Synthesis
Ardkhean, R., Caputo, D. F. J., Morrow, S. M., Shi H., Xiong, Y and Anderson, E. A.
Chem. Soc. Rev. 2016, 45, 1557.

2. Strategic Application and Transformation of ortho-Disubstituted Phenyl and Cyclopropyl Ketones to Expand the Scope of Hydrogen Borrowing Catalysis
Frost, J. R., Cheong, C. B., Akhtar, W. M., Caputo, D. F. J., Stevenson, N. G. and Donohoe, T. J.
J. Am. Chem. Soc. 2015, 137, 15664.

1. Active-Metal Template Synthesis of a Halogen-Bonding Rotaxane for Anion Recognition
Langton, M. J., Xiong, Y. and Beer, P. D.
Chem. Eur. J. 2015, 21, 18910.