PUBLICATIONS

Our students have published their research in a wide variety of high-impact scientific journals. Please see below a list of all SBM CDT research publications.

Preprints
P8. Stereoselective Alder-ene Reactions of Bicyclo[1.1.0]butanes: Facile Synthesis of Cyclopropyl- and Aryl-substituted Cyclobutenes.
Dasgupta, A., Bhattacharjee, S., Tong, Z., Guin, A., McNamee, R., Christensen, K., Biju, A. and Anderson, E. A.
ChemRxiv, 2023, Preprint.
P7. Studies on the selectivity of the SARS-CoV-2 papain-like protease reveal the importance of the P2' proline of the viral polyprotein.
Chan, H. H. T, Brewitz, L., Strain-Damerell, C., Lukacik, P., Walsh, M. A., Schofield, C. J. and Duarte, F.
bioRxiv, 2023, Preprint.
P6. A radical-polar crossover approach to complex nitrogen heterocycles via the triplet state.
Lockhart, Z., Popescu, M., Alegre-Requena, J., Ahuja, J, Paton, R. and Smith, M. D.
ChemRxiv, 2023, Preprint.
P5. 1,2-Redox Transpositions of Tertiary Amides.
Shennan, B., Sanchez Alonso, S. and Dixon, D. J.
ChemRxiv, 2023, Preprint.
P3. Harnessing triaryloxonium ions for aryne generation.
Smith, O., Hindson, M., Sreenithya, A., Tataru, V., Paton, R., Burton, J. and Smith, M. D.
ChemRxiv, 2023, Preprint.
P2. Taming non-classical carbocations to control small ring reactivity.
McNamee, R. E., Frank, N., Christensen, K, Duarte, F. and Anderson, E. A.
ChemRxiv, 2023, Preprint.
P1. Intact nucleosomal context enables chromodomain reader MRG15 to distinguish H3K36me3 from -me2.
Faulkner, S., Couturier, A. M., Josephson, B., Watts, T., Davis, B. G. and Esashi, F.
bioRxiv, 2020, Preprint.

2023
265. Fluorochemicals from fluorspar via a phosphate-enabled mechanochemical process that bypasses HF.
Patel, C., André-Joyaux, E., Leitch, J. A., Martínez De Irujo-Labalde, X., Ibba, F., Struijs, J., EllWanger, M. A., Paton, R., Browne, D. L., Pupo, G., Aldridge, S., Hayward, M. A. and Gouverneur, V.
Science, 2023, 381, 302.
Stacks Image 10243
264. Synthesis of Cyclopropanes via Hydrogen-Borrowing Catalysis.
Crompton, J. L., Frost, J. R., Rowe, S. M., Christensen, K. E. and Donohoe, T. J.
Org. Lett., 2023, 25, 5253.
Stacks Image 10575
263. Engineering cellular communication between light-activated synthetic cells and bacteria.
Smith, J. M., Hartmann, D. and Booth, M. J.
bioRxiv, 2022, Preprint.
Nat. Chem. Biol.,
2023, Accepted Article.
Stacks Image 10363
262. Redox Reorganization: Aluminium Promoted 1,5-Hydride Shifts Allow the Controlled Synthesis of Multisubstituted Cyclohexenes.
Smith, L., Armstrong, R., Hou, J., Smith, E., Sze, M., Sterling, A., Smith, A., Duarte, F. and Donohoe, T. J.
Angew. Chem. Int. Ed., 2023, Early View.
Stacks Image 10557
261. Solution-processable polymers of intrinsic microporosity for gas-phase carbon dioxide photoreduction.
Moruzzi, F., Zhang, W., Purushothaman, B., Gonzalez-Carrero, S., Aitchison, C., Willner, B., Ceugniet, F., Lin, Y., Kosco, J., Chen, H., Tian, J., Alsufyani, M, Gibson, J., Rattner, E., Baghdadi, Y., Eslava, S., Neophytou, M., Durrant, J., Steier, L. & McCulloch, I.
Nat. Commun., 2023, 14, 3443.
260. Dynamical nonequilibrium molecular dynamics simulations identify allosteric sites and positions associated with drug resistance in the SARS-CoV-2 main protease.
Chan, H.T.H., Oliveira, A.S.F., Schofield, C.J., Mulholland, A.J. and Duarte, F.
bioRxiv, 2022, Preprint.
JACS Au,
2023, 3, 1767.
Stacks Image 10545
259. A general scheme for generating NMR supersequences combining high- and low-sensitivity experiments.
Yong, J.R.J., Kupčeb E. and Claridge, T.D.W.
Chem. Commun., 2023, 59, 7827.
Stacks Image 10539
258. Templated 2D Polymer Heterojunctions for Improved Photocatalytic Hydrogen Production.
Aitchison, C.M., Gonzalez- Carrero, S., Yao, S., Benkert, M., Ding, Z., Young, N.P., Willner, B., Moruzzi, F., Lin, Y., Tian, J., Nellist, P.D., Durrant, J.R. and McCulloch, I.
Adv. Mater., 2023, Early View.
Stacks Image 10533
257. Catalytic Enantioselective Intramolecular Oxa-Michael Reaction to α,β-Unsaturated Esters and Amides.
Su, G., Formica, M., Yamazaki, K., Hamlin, T. A. and Dixon, D. J.
J. Am. Chem. Soc., 2023, 145, 12771.
Stacks Image 10357
256. Catalytic Enantioselective Nucleophilic Desymmetrisation of Phosphonate Esters.
Formica, M., Rogova, T., Shi, H., Sahara, N., Ferko, B., Farley, A., Christensen, K., Duarte, F., Yamazaki, K. and Dixon, D. J.
ChemRxiv, 2021, Preprint.
Nature Chem.,
2023, 15, 714.
Stacks Image 10521
255. Orthogonal Light-Activated DNA for Patterned Biocomputing within Synthetic Cells.
Hartmann, D., Chowdhry, R., Smith, J. and Booth, M.
ChemRxiv, 2022, Preprint.
J. Am. Chem. Soc.,
2023, 145, 9471.
Stacks Image 10375
254. Precise, Orthogonal Remote-Control of Cell-Free Systems Using Photocaged Nucleic Acids.
Mazzotti, G., Hartmann, D. and Booth, M.
ChemRxiv, 2023, Preprint.
J. Am. Chem. Soc.,
2023, 145, 9481.
Stacks Image 10427
253. Cyclic peptides target the aromatic cage of a PHD-finger reader domain to modulate epigenetic protein function.
Coleman, O. D., Macdonald, J., Thomson, B., Ward, J. A., Stubbs, C. J., McAllister, T. E., Clark, S., Amin, S., Cao, Y., Abboud, M. I., Zhang, Y, Sanganee, H., Huber, K. V. M. Claridge, T. D. W. and Kawamura, A.
Chem. Sci., 2023, 14, 7136.
Stacks Image 10411
252. Handcuffed antisense oligonucleotides for light-controlled cell-free expression.
Hartmann, D. and Booth, M.
Chem. Commun., 2023, 59, 5685.
Stacks Image 10509
251. Accessible light-controlled knockdown of cell-free protein synthesis using phosphorothioate-caged antisense oligonucleotides.
Hartmann, D. and Booth, M.
ChemRxiv, 2022, Preprint.
Commun. Chem.,
2023, 6, 59.
Stacks Image 10485
250. A photoswitchable solvatochromic dye for probing membrane ordering by RESOLFT super-resolution microscopy.
Frawley, A., Leslie, K., Wycisk, V., Galiani, S., Shrestha, D., Eggeling, C. and Anderson, H. L.
ChemRxiv, 2023, Preprint.
ChemPhysChem,
2023, 24, e202300125.
Stacks Image 10473
249. Kinetic and inhibition studies on human Jumonji-C (JmjC) domain-containing protein 5.
Tumber, A., Salah, E., Brewitz, L., Corner, T. P. and Schofield, C. J.
RSC Chem. Biol., 2023, 4, 399.
Stacks Image 10417
248. Mobile Molecules: Reactivity Profiling Guides Faster Movement on a Cysteine Track.
Bo, Z., Lim, Z. H., Duarte, F., Bayley, H., Qing, Y.
Angew. Chem. Int. Ed., 2023, 62, e202300890.
Stacks Image 10497
247. Bifunctional Iminophosphorane-Catalyzed Enantioselective Nitroalkane Addition to Unactivated α,β-Unsaturated Esters.
Rozsar, D., Farley, A., McLauchlan, I., Shennan, B. A., Yamazaki, K. and Dixon, D. J.
ChemRxiv, 2022, Preprint.
Angew. Chem. Int. Ed.,
2023, 62, e202303391.
Stacks Image 10467
246. Control of stereogenic oxygen in a helically chiral oxonium ion.
Smith, O., Popescu, M., Hindson, M., Paton, R., Burton, J. and Smith, M. D.
ChemRxiv, 2022, Preprint.
Nature,
2023, 615, 430.
Stacks Image 10369
245. Visible Light Photoredox-Catalyzed Decarboxylative Alkylation of 3-Aryl-Oxetanes and Azetidines via Benzylic Tertiary Radicals and Implications of Benzylic Radical Stability.
Dubois, M. A. J., Rojas, J. J., Sterling, A. J., Broderick, H. C., Smith, M. A., White, A. J. P., Miller, P. W., Choi, C., Mousseau, J. J., Duarte, F. and Bull, J. A.
J. Org. Chem.,
2023, 88, 6476.
Stacks Image 10456
244. Stereoretentive Post-Translational Protein Editing.
Fu, X-P., Yuan, Y., Jha, A., Levin, N., Giltrap, A. M., Ren, J., Mamalis, D., Mohammed, S. and Davis, B. G.
ACS Cent. Sci.,
2023, 9, 405.
Stacks Image 10453
243. Enantioselective Total Synthesis of (−)-Himalensine A via a Palladium and 4-Hydroxyproline Co-catalyzed Desymmetrization of Vinyl-bromide-tethered Cyclohexanones.
Kučera, R., Ellis, S. E., Yamazaki, K., Hayward Cooke, J., Chekshin, N., Christensen, K. E., Hamlin, T. A. and Dixon, D. J.
J. Am. Chem. Soc.,
2023, 145, 5422.
Stacks Image 10479
242. Catalytic enantioselective 6𝝿 photocyclization of acrylanilides
Jones, B., Solon, P., Popescu, M., Du, J.-Y., Paton, R. and Smith, M. D.
ChemRxiv, 2022, Preprint.
J. Am. Chem. Soc.,
2023, 145, 171.
Stacks Image 10439
241. Enantioselective synthesis of atropisomeric indoles via iron-catalysed oxidative cross-coupling
Surgenor, R., Liu, X., Keenlyside, M., Myers, W. and Smith M. D.
ChemRxiv, 2021, Preprint.
Nat. Chem.,
2023, 15, 357.
Stacks Image 10005
240. Alcohols as efficient intermolecular initiators for a highly stereoselective polyene cyclisation cascade.
Aynetdinova, D., Jacques, R., Christensen, K. and Donohoe, T. J.
Chem. Eur. J., 2023, 29, e202203732.
Stacks Image 10399

2022
239. Total Synthesis and Structure Confirmation of (E) and (Z)-Ocellenyne.
Hicks, H. B., Brown, D. S., Chan, H. S. S., Sousa, B. A., Christensen, K. E. and Burton, J. W.
Org. Lett., 2022, 24, 9174.
Stacks Image 10321
238. Photo-switchable anion binding and catalysis with a visible light responsive halogen bonding receptor.
Kerckhoffs, A., Moss, I. and Langton, M. J.
Chem. Commun., 2023, 59, 51.
Stacks Image 10393
237. Recent advances in the dearomative functionalisation of heteroarenes.
Kratena, N., Marinic, B. and Donohoe, T. J.
Chem. Sci., 2022, 13, 14213.
Stacks Image 10387
236. Rapid and scalable halosulfonylation of strain-release reagents.
Pickford, H. D., Ripenko, V., McNamee, R. E., Holovchuk, S., Thompson, A. L., Smith, R. C., Mykhailiuk, P. K. and Anderson, E. A.
ChemRxiv, 2022, Preprint.
Angew. Chem. Int. Ed.,
2023, 62, e202213508.
Stacks Image 10381
235. Rhodium-Catalyzed [2 + 2 + 2] Cyclotrimerizations of Yndiamides with Alkynes.
Smith, P. J., Tong, Z., Ragus, J., Solon, P., Shimkin, K. W. and Anderson, E. A.
Org. Lett., 2022, 24, 7522.
Stacks Image 10351
234. Enantioselective oxidation of unactivated C–H bonds in cyclic amines by iterative docking-guided mutagenesis of P450BM3 (CYP102A1).
Zhang, Y., Xiong, Z., Li, Y., Wilson, M., Christensen, K. E., Jaques, E., Hernández-Lladó, P., Robertson, J. and Wong, L. L.
Nat. Synth.,
2022, 1, 936.
Stacks Image 10345
232. Synthesis of meta-substituted arene bioisosteres from [3.1.1]propellane.
Frank, N., Nugent, J., Shire, B.R., Pickford, H. D., Rabe, P., Sterling, A. J., Zarganes-Tzitzikas, T., Grimes, T., Thompson, A. L., Smith, R. C., Schofield, C. J., Brennan, P. E., Duarte, D. and Anderson, E. A.
ChemRxiv, 2022, Preprint.
Nature,
2022, 611, 721.
231. Identification of Histone Peptide Binding Specificity and Small-Molecule Ligands for the TRIM33α and TRIM33β Bromodomains.
Sekirnik, A., Reynolds, J., See, L., Bluck, J., Scorah, A., Tallant, C., Lee, B., Leszczynska, K., Grimley, R., Storer, R. I., Malattia, M, Crespillo, S., Caria, S., Duclos, S., Hammond, E. M., Knapp, S., Morris, G. M., Duarte, F., Biggin, P., and Conway, S. J.
ChemRxiv, 2022, Preprint.
ACS Chem. Biol.,
2022, 17, 2753.
Stacks Image 10327
229. Towards fully optimised and automated ESR spectroscopy.
Verstraete, J.-B., Yong, J. R. J., Goodwin, D. L., Myers, W. K. and Foroozandeh, M.
Chem. Commun., 2022, 58, 10715.
Stacks Image 10315
228. A Vicinal Diol Approach for the Total Synthesis of Molestin E, ent-Sinulacembranolide A and ent-Sinumaximol A.
Hoff, O., Kratena, N., Aynetdinova, D., Christensen, K. E. and Donohoe, T. J.
Chem. Eur. J., 2022, 28, e202202464.
Stacks Image 10309
227. Counterion-Mediated Enantioconvergent Synthesis of Axially Chiral Medium Rings.
Du, J.-Y., Balan, T., Claridge, T. D. W. C and Smith, M. D.
J. Am. Chem. Soc., 2022, 144, 14790.
Stacks Image 10303
226. N-Sulfinyl-O-(tert-Butyl)Hydroxylamine.
Davies, T. Q. and Willis, M. C.
In Encyclopedia of Reagents for Organic Synthesis. John Wiley & Sons, 2022.
Stacks Image 10238
225. An LNA-amide modification that enhances the cell uptake and activity of phosphorothioate exon-skipping oligonucleotides.
Baker, Y.R., Thorpe, C., Chen, J., Poller, L. M., Cox, L., Kumar, P., Lim, W. F., Lie, L., McClorey, G., Epple, S., Singleton, D., McDonough, M. A., Hardwick, J. S., Christensen, K. E., Wood, M. J. A., Hall, J. P., El-Sagheer, A. H., and Brown, T.
Nat. Commun., 2022, 13, 4036.
224. Alcohols as Alkylating Agents in the Cation-Induced Formation of Nitrogen Heterocycles.
Cox, L., Zhu, Y., Smith, P. J., Christensen, K. E., Sidera Portela, M. and Donohoe, T. J.
Angew. Chem. Int. Ed., 2022, 61, e202206800.
Stacks Image 10285
223. Branching out: redox strategies towards the synthesis of acyclic α-tertiary ethers.
Shennan, B. D. A., Berheci, D., Crompton, J. L., Davidson, T. A., Field, J. L., Williams, B. A and Dixon, D. J.
Chem. Soc. Rev., 2022, 51, 5878.
Stacks Image 10279
222. Modular Two-Step Route to Sulfondiimidamides.
Zhang, Z.-X., Bell, C., Ding, M. and Willis, M. C.
J. Am. Chem. Soc., 2022, 144, 11851.
Stacks Image 10273
221. An autonomously oscillating supramolecular self-replicator.
Howlett, M.G., Engwerda, A.H.J., Scanes, R.J.H. and Fletcher, S. P.
Nat. Chem., 2022, 14, 805.
Stacks Image 10267
220. Evolution of the Dearomative Functionalization of Activated Quinolines and Isoquinolines: Expansion of the Electrophile Scope.
Kischkewitz, M., Marinic, B., Kratena, N., Lai, Y., Hepburn, H. B., Dow, M., Christensen, K. E. and Donohoe,T. J.
Angew. Chem. Int. Ed., 2022, 61, e202204682.
Stacks Image 10261
219. Photocatalytic Late- Stage Functionalization of Sulfonamides via Sulfonyl Radical Intermediates.
Tilby, M.J ., Dewez, D. F., Pantaine, L. R. E., Hall, A., Martínez-Lamenca, C. and Willis, M. C.
ACS Catal., 2022, 12, 6060.
Stacks Image 10255
218. Extension of hydrogen borrowing alkylation reactions for the total synthesis of (−)-γ-lycorane.
Hall, C., Marriott, I., Christensen, K., Day, A., Goundry, W. and Donohoe, T. J.
Chem. Commun., 2022, 58, 4966.
Stacks Image 10249
217. [18F]Difluorocarbene for Positron Emission Tomography.
Sap, J.B.I., Meyer, C.F., Ford, J., Straathof, N., Dürr, A., Lelos, M., Paisey, S., Mollner, T., Hell, S., Trabanco, A., Genicot, C., am Ende, C., Paton, R. S., Tredwell, M. and Gouverneur, V..
Nature, 2022, 606, 102.
216. Transition Metal-Free, Visible Light-Mediated Radical Cyclisation of Malonyl Radicals onto 5-Ring Heteroaromatics.
Hernández-Lladó, P., Garrec, K., Schmitt, D. and Burton, J.
Adv. Synth. Catal., 2022, 364, 1724.
Stacks Image 10229
215. Reading and erasing of the phosphonium analogue of trimethyllysine by epigenetic proteins.
Kamps, J.J.A.G., Belle, R., Poater, J., Kumar, K., Pieters, B., Salah, E., Claridge, T. D. W., Paton, R., S., Bickelhaupt, F. M., Kawamura, A., Schofield, C. J. and Mecinović, J.
Commun. Chem., 2022, 5, 27.
Stacks Image 10223
214. Asymmetric Azidation under Hydrogen Bonding Phase-Transfer Catalysis: A Combined Experimental and Computational Study.
Wang, J., Horwitz, M. A., Dürr, A. B., Ibba, F., Pupo, G., Gao, Y., Ricci, P., Christensen, K. E., Pathak, T. P., Claridge, T. D. W. C., Lloyd-Jones, G. C., Paton, R. S. and Gouverneur, V.
J. Am. Chem. Soc., 2022, 144, 4572.
Stacks Image 10217
213. A Silyl Sulfinylamine Reagent Enables the Modular Synthesis of Sulfonimidamides via Primary Sulfinamides.
Ding, M., Zhang, Z.-X., Davies, T. Q. and Willis, M. C.
Org. Lett., 2022, 24, 1711.
Stacks Image 10211
212. Amino-oxetanes as amide isosteres by an alternative defluorosulfonylative coupling of sulfonyl fluorides.
Rojas, J. J., Croft, R. A., Sterling, A. J., Briggs, E. L., Antermite, D., Schmitt, D., Blagojevic, L., Haycock, P., White, A., Duarte, F., Choi, C., Mousseau, J. and Bull, J. A.
Nat. Chem., 2022, 14, 160.
Stacks Image 10203
211. DABSO – A Reagent to Revolutionize Organosulfur Chemistry.
Andrews, J. A. and Willis, M. C.
Synthesis, 2022, 54, 1695.
Stacks Image 10197
210. Modular Pulse Program Generation for NMR Supersequences.
Yong, J. R. J., Kupce, E. and Claridge, T. D. W.
Anal. Chem., 2022, 94, 2271.
Stacks Image 10191
209. Diverse saturated heterocycles from a hydroacylation/conjugate addition cascade.
Iwumene, N. U. N., Moseley, D. F., Pullin, R. C. and Willis, M. C.
Chem. Sci., 2022, 13, 1504.
Stacks Image 10180
208. Characterisation of the SARS-CoV-2 ExoN (nsp14ExoN-nsp10) complex: implications for its role in viral genome stability and inhibitor identification.
Baddock, H., Brolih, S., Yosaatmadja, Y., Ratnaweera, M., Bielinski, M., Swift, L., Cruz-Migoni, A., Fan, H., Keown, J., Walker, A., Morris, G. M., Grimes, J., Fodor, E., Schofield, C. J., Gileadi, O. and McHugh, P. J.
bioRxiv, 2020, Preprint.
Nucleic Acids Res.,
2022, 50, 1484.
207. A New Organocatalytic Desymmetrization Reaction Enables the Enantioselective Total Synthesis of Madangamine E.
Shiomi, S., Shennan, B., Yamazaki, K., Fuentes de Arriba, Á.L., Vasu, D., Hamlin, T. A. and Dixon, D. J.
ChemRxiv, 2021, Preprint.
J. Am. Chem. Soc.,
2022, 144, 1407.
Stacks Image 10177
206. Bifunctional Iminophosphorane-Catalyzed Enantioselective Sulfa-Michael Addition to Unactivated α,β-Unsaturated Amides.
Rozsar, D., Formica, M., Yamazaki, K., Hamlin, T. and Dixon, D. J.
ChemRxiv, 2021, Preprint.
J. Am. Chem. Soc.,
2022, 144, 1006.
Stacks Image 9885

2021
205. Synthesis and Applications of Polysubstituted Bicyclo[1.1.0]butanes.
McNamee, R. E.
, Thompson, A. L. and Anderson E. A.
J. Am. Chem. Soc., 2021, 143, 21246.
Stacks Image 10143
204. Synthesis and Application of Constrained Amidoboronic Acids Using Amphoteric Boron-Containing Building Blocks.
Soor, H. S., Diaz, D. B., Tsui, K. Y., Calvopiña, K., Bielinski, M., Tantillo, D. J., Schofield, C. J. and Yudin, A. K.
J. Org. Chem., 2022, 87, 94.
Stacks Image 10171
203. Single photon double and triple ionization of allene.
Ideböhn, V., Sterling, A. J., Wallner, M., Olsson, E., Squibb, R. J., Miniotaite, U., Forsmalm, E., Forsmalm, M., Stranges, S., Dyke, J. M., Duarte, F., Eland, J. H. D., and Feifel, R.
Phys. Chem. Chem. Phys., 2022, 24, 786.
Stacks Image 10161
202. First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53.
Nowak, R., Tumber, A., Hendrix, E., Ansari, M., Sabatino, M., Antonini, L., Andrijes, R., Salah, E., Mautone, N., Pellegrini, F., Simelis, K., Kawamura, A., Johansson, C., Passeri, D., Pellicciari, R., Ciogli, A., Del Bufalo, D., Ragno, R., Coleman, M., Trisciuoglio, D., Mai, A., Oppermann, U., Schofield, C. J. and Rotili, D.
J. Med. Chem., 2021, 64, 17031.
Stacks Image 10149
201. Lactone Backbone Density in Rigid Electron-Deficient Semiconducting Polymers Enabling High n-type Organic Thermoelectric Performance.
Alsufyani, M., Stoeckel, M.-A., Chen, X., Thorley, K., Hallani, R.K., Puttisong, Y., Ji, X., Meli, D., Paulsen, B.D., Strzalka, J., Regeta, K., Combe, C., Chen, H., Tian, J., Rivnay, J., Fabiano, S. and McCulloch, I.
Angew. Chem. Int. Ed., 2022, 61, e202113078.
Stacks Image 10155
200. Parallel NMR Supersequences: Ten Spectra in a Single Measurement.
Kupče, E., Yong, J. R. J., Widmalm, G. and Claridge, T. D. W.
JACS Au, 2021, 1, 1892.
Stacks Image 10131
199. Electrophilic Activation of [1.1.1]Propellane for the Synthesis of Nitrogen-Substituted Bicyclo[1.1.1]pentanes.
Livesley, S., Sterling, A.J., Robertson, C.M., Goundry, W.R.F., Morris, J.A., Duarte, F. and Aïssa, C.
Angew. Chem. Int. Ed., 2022, 61, e202111291.
Stacks Image 10137
198. Benzenemethanamine, α,α-Diphenyl-N-Sulfinyl-.
Tilby, M. and Willis, M. C.
In Encyclopedia of Reagents for Organic Synthesis. John Wiley & Sons, 2021.
Stacks Image 10125
197. Synthesis of α-Quaternary Bicyclo[1.1.1]pentanes through Synergistic Organophotoredox and Hydrogen Atom Transfer Catalysis.
Nugent, J., Sterling, A. J., Frank, N., Mousseau, J. J. and Anderson, E. A.
Org. Lett., 2021, 23, 8628.
Stacks Image 10101
196. Sulfinates from Amines: A Radical Approach to Alkyl Sulfonyl Derivatives via Donor–Acceptor Activation of Pyridinium Salts.
Andrews, J., Pantaine, L., Palmer, C. F., Poole, D. L. and Willis, M. C.
Org. Lett., 2021, 23, 8488.
Stacks Image 10119
195. A Three-Component Ugi-Type Reaction of N-Carbamoyl Imines Enables a Broad Scope Primary α-Amino 1,3,4-Oxadiazole Synthesis.
Matheau-Raven, D., Boulter, E., Rogova, T. and Dixon, D. J.
Org. Lett., 2021, 23, 8209.
Stacks Image 10107
194. Red-shifted tetra-ortho-halo-azobenzenes for photo-regulated transmembrane anion transport.
Kerckhoffs, A., Bo, Z., Penty, S. E., Duarte, F. and Langton, M. J.
Org. Biomol. Chem., 2021, 19, 9058.
Stacks Image 9981
193. Exploiting Configurational Lability in Aza-Sulfur Compounds for the Organocatalytic Enantioselective Synthesis of Sulfonimidamides.
Tilby, M. J., Dewez, D. F., Hall, A., Martínez Lamenca, C. and Willis, M. C.
Angew. Chem. Int. Ed., 2021, 60, 25680.
Stacks Image 10095
192. A New 1,5-Disubstituted Triazole DNA Backbone Mimic with Enhanced Polymerase Compatibility.
Epple, S., Modi, A., Baker, Y. R., Wȩgrzyn, E., Traoré, D., Wanat, P., Tyburn, A., Shivalingam, A., Taemaitree, L., El-Sagheer, A. and Brown, T.
J. Am. Chem. Soc., 2021, 143, 16293.
Stacks Image 10089
191. Azine-N-oxides as effective controlling groups for Rh-catalysed intermolecular alkyne hydroacylation.
Moseley, D. F., Kalepua, J. and Willis, M. C.
Chem. Sci., 2021, 12, 13068.
Stacks Image 10083
190. Discovery of SARS-CoV-2 Mpro Peptide Inhibitors from Modelling Substrate and Ligand Binding.
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ACS Catal. 2017, 7, 6587.
Stacks Image 8729
19. Exploiting Carbonyl Groups to Control Intermolecular Rhodium-Catalyzed Alkene and Alkyne Hydroacylation
Coxon, T. J., Fernandez, M., Barwick-Silk, J., McKay, A. I., Britton, L. E., Weller, A. S., Willis, M. C.
J. Am. Chem. Soc. 2017, 139, 10142.
Stacks Image 8749
18. Visible light photocatalysis of 6π heterocyclization
Münster, N., Parker, N. A., van Dijk, L., Paton, R. S., Smith, M. D.
Angew. Chem. Int. Ed. 2017, 56, 9468.
Stacks Image 8743
17. Unexpected Interactions between Alkyl Straps and Pyridine Ligands in Sulfur-Strapped Porphyrin Nanorings
Roche, C., Lou, Q., Gil-Ramirez, G., Jiang, H.-W., Kohn, D. R., Xiong, Y., Thompson, A. L., Anderson, H. L.
J. Org. Chem. 2017, 82, 7446.
Stacks Image 8761
16. Potential for minimal self-replicating systems in a dynamic combinatorial library of equilibrating imines
Morrow, S. M.
, Bissette, A. J., Fletcher, S. P.
Tetrahedron 2017, 73, 5005.
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15. Transmission of chirality through space and across length scales
Morrow, S. M.
, Bissette, A. J. and Fletcher, S. P.
Nature Nanotechnology 201712, 410.
Stacks Image 8755
14. Structural and stereoelectronic insights into oxygenase-catalyzed formation of ethylene from 2-oxoglutarate
Zhang, Z., Smart, T. J., Choi, H., Hardy, F., Lohansa, C. T., Abboud, M. I., Richardson, M. S. W., Paton, R. S., McDonough, M. A. and Schofield, C. J.
Proc. Natl. Acad. Sci. 2017, 114, 4667. 
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13. Neutral iodotriazole foldamers as tetradentate halogen bonding anion receptors
Borissov, A.
, Lim, J. Y. C., Brown, A., Christensen, K. E., Thompson, A. L., Smith, M. D. and Beer, P. D.
Chem. Commun. 2017, 53, 2483.
Stacks Image 8781
12. Discovery of a PCAF Bromodomain Chemical Probe
Moustakim, M.
, Clark, P. G. K., Trulli, L., Fuentes de Arriba, A. L., Ehebauer, M. T., Chaikuad, A., Murphy, E. J., Mendez-Johnson, J., Daniels, D., Hou, C.-F. D., Lin, Y.-H., Walker, J. R., Hui, R., Yang, H., Dorrel, L., Rogers, C. M., Monteiro, O. P., Fedorov, O., Huber, K. V. M., Knapp, S., Heer, J., Dixon, D. J., Brennan, P. E.
Angew. Chem. Int. Ed. 201756, 827. DOI: 10.1002/anie.201610816.
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2016
10. A Cascade Strategy Enables a Total Synthesis of (+/-)-Morphine
Chu, S., Münster, N., Balan, T., Smith. M. D.
Angew. Chem. Int. Ed. 2016, 55, 14306.
Stacks Image 8807
9. Posttranslational mutagenesis: A chemical strategy for exploring protein side-chain diversity
Wright, T. H., Bower, B. J., Chalker, J. M., Bernardes, G. J. L., Wiewiora, R., Ng, W.-L., Raj, R., Faulkner, S., Vallée, M. R. J., Phanumartwiwath, A., Coleman, O. D., Thézénas, M.-L., Khan, M., Galan, S. R. G., Lercher, L., Schombs, M. W., Gerstberger, S., Palm-Espling, M. E., Baldwin, A. J., Kessler, B. M., Claridge, T. D. W., Mohammed, S. and Davis, B. G.
Science 2016, 354, 597.
Stacks Image 8813
8. Chemical Probes and Inhibitors of Bromodomains outside the BET family
Moustakim, M.
, Clark, P. G. K., Hay, D. A., Dixon, D. J. and Brennan, P. E.
Med. Chem. Commun. 2016, 7, 2246.
Stacks Image 8819
7. Photoswitchable Spiropyran Dyads for Biological Imaging
Xiong, Y.
, Rivera-Fuentes, P., Sezgin, E., Jentzsch, A. V., Eggeling, C. and Anderson, H. L.
Org. Lett. 2016, 8, 3666.
Stacks Image 8825
6. Cp2ZrMeCl: A Reagent for Asymmetric Methyl Addition
Garrec, K
. and Fletcher, S. P.
Org. Lett. 2016, 8, 3814.
Stacks Image 8831
5. Recent Applications in Natural Product Synthesis of Dihydrofuran and -pyran Formation by Ring-closing Alkene Metathesis
Jacques, R.
, Pal, R., Parker, N. A., Sear, C. E., Smith, P. W., Ribaucourt, A. and Hodgson, D. M.
Org. Biomol. Chem. 2016, 14, 5875.
Stacks Image 8837
4. Organocatalytic Enantioselective Desymmetrisation
Borissov, A.
, Davies, T. Q., Ellis, S. R., Fleming T. F., Richardson, M. S. W. and Dixon, D. J.
Chem. Soc. Rev. 2016, 45, 5474.
Stacks Image 8843
3. Cascade Polycyclizations in Natural Product Synthesis
Ardkhean, R.
, Caputo, D. F. J., Morrow, S. M., Shi H., Xiong, Y and Anderson, E. A.
Chem. Soc. Rev. 2016, 45, 1557.
Stacks Image 8787

2015
2. Strategic Application and Transformation of ortho-Disubstituted Phenyl and Cyclopropyl Ketones to Expand the Scope of Hydrogen Borrowing Catalysis
Frost, J. R., Cheong, C. B., Akhtar, W. M., Caputo, D. F. J., Stevenson, N. G. and Donohoe, T. J.
J. Am. Chem. Soc. 2015, 137, 15664.
Stacks Image 8855
1. Active-Metal Template Synthesis of a Halogen-Bonding Rotaxane for Anion Recognition
Langton, M. J., Xiong, Y. and Beer, P. D.
Chem. Eur. J. 2015, 21, 18910.
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Stacks Image 8654
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