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P3. Enantioselective synthesis of atropisomeric indoles via iron catalysed oxidative cross-coupling.
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P2. Characterisation of the SARS-CoV-2 ExoN (nsp14^ExoN-nsp10) complex: implications for its role in viral genome stability and inhibitor identification.
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P1. Intact nucleosomal context enables chromodomain reader MRG15 to distinguish H3K36me3 from -me2.
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208. Diverse saturated heterocycles from a hydroacylation/conjugate addition cascade.
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207. A New Organocatalytic Desymmetrization Reaction Enables the Enantioselective Total Synthesis of Madangamine E.
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206. Bifunctional Iminophosphorane-Catalyzed Enantioselective Sulfa-Michael Addition to Unactivated α,β-Unsaturated Amides.
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205. Synthesis and Applications of Polysubstituted Bicyclo[1.1.0]butanes.
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204. Synthesis and Application of Constrained Amidoboronic Acids Using Amphoteric Boron-Containing Building Blocks.
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203. Single photon double and triple ionization of allene.
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202. First-in-Class Inhibitors of the Ribosomal Oxygenase MINA53.
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201. Lactone Backbone Density in Rigid Electron-Deficient Semiconducting Polymers Enabling High n-type Organic Thermoelectric Performance.
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200. Parallel NMR Supersequences: Ten Spectra in a Single Measurement.
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199. Electrophilic Activation of [1.1.1]Propellane for the Synthesis of Nitrogen-Substituted Bicyclo[1.1.1]pentanes.
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198. Benzenemethanamine, α,α-Diphenyl-N-Sulfinyl-.
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197. Synthesis of α-Quaternary Bicyclo[1.1.1]pentanes through Synergistic Organophotoredox and Hydrogen Atom Transfer Catalysis.
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196. Sulfinates from Amines: A Radical Approach to Alkyl Sulfonyl Derivatives via Donor–Acceptor Activation of Pyridinium Salts.
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195. A Three-Component Ugi-Type Reaction of N-Carbamoyl Imines Enables a Broad Scope Primary α-Amino 1,3,4-Oxadiazole Synthesis.
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194. Red-shifted tetra-ortho-halo-azobenzenes for photo-regulated transmembrane anion transport.
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193. Exploiting Configurational Lability in Aza-Sulfur Compounds for the Organocatalytic Enantioselective Synthesis of Sulfonimidamides.
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192. A New 1,5-Disubstituted Triazole DNA Backbone Mimic with Enhanced Polymerase Compatibility.
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191. Azine-N-oxides as effective controlling groups for Rh-catalysed intermolecular alkyne hydroacylation.
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190. Discovery of SARS-CoV-2 Mpro Peptide Inhibitors from Modelling Substrate and Ligand Binding.
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189. Regio- and stereoselective addition of Brønsted acids to yndiamides: Synthesis of N,O,N- and N,S,N-trisubstituted ketene acetals.
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188. Switchable, Reagent-Controlled Diastereodivergent Photocatalytic Carbocyclisation of Imine-Derived α-Amino Radicals.
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187. X-ray free-electron laser studies reveal correlated motion during isopenicillin N synthase catalysis.
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186. Selection between Competing Self-Reproducing Lipids: Succession and Dynamic Activation.
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185. A phosphate binding pocket is a key determinant of exo- versus endo-nucleolytic activity in the SNM1 nuclease family.
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184. Structural and mechanistic insights into the Artemis endonuclease and strategies for its inhibition.
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183. Synthesis of Polysubstituted Fused Pyrroles by Gold-Catalyzed Cycloisomerization/1,2-Sulfonyl Migration of Yndiamides.
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182. Base-Activated Latent Heteroaromatic Sulfinates as Nucleophilic Coupling Partners in Palladium-Catalyzed Cross-Coupling Reactions.
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181. On-the-Fly, Sample-Tailored Optimization of NMR Experiments.
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180. Supramolecular chemistry in lipid bilayer membranes.
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179. Artificial nucleic acid backbones and their applications in therapeutics, synthetic biology and biotechnology.
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178. An on-demand, drop-on-drop method for studying enzyme catalysis by serial crystallography.
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177. A General Iridium-Catalyzed Reductive Dienamine Synthesis Allows a Five-Step Synthesis of Catharanthine via the Elusive Dehydrosecodine.
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176. Controlling Intramolecular Interactions in the Design of Selective, High-Affinity, Ligands for the CREBBP Bromodomain.
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175. How do we address neglected sulfur pharmacophores in drug discovery?
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174. A catalytic asymmetric cross-coupling approach to the synthesis of cyclobutanes.
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173. General α-Amino 1,3,4-Oxadiazole Synthesis via Late-Stage Reductive Functionalization of Tertiary Amides and Lactams.
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172. Twofold Radical-Based Synthesis of N,C-Difunctionalized Bicyclo[1.1.1]pentanes.
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171. Increasing Sensitivity and Versatility in NMR Supersequences with New HSQC-based Modules.
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170. Rh-catalyzed asymmetric Suzuki-Miyaura cross-coupling.
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169. General Pyrrolidine Synthesis via Iridium-Catalyzed Reductive Azomethine Ylide Generation from Tertiary Amides and Lactams.
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168. Au(I)-Catalyzed Oxidative Functionalization of Yndiamides.
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167. Late-stage difluoromethylation: concepts, developments and perspective.
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166. Highly Active Halogen Bonding and Chalcogen Bonding Chloride Transporters with Non-Protonophoric Activity.
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165. Acceleration of lipid reproduction by emergence of microscopic motion.
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164. Synthesis of 1,3-disubstituted bicyclo[1.1.0]butanes via directed bridgehead functionalization.
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163. Rediscovering Sulfinylamines as Reagents for Organic Synthesis.
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162. A Novel Automated Screening Method For Combinatorial Small Molecules.
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161. Parallel nuclear magnetic resonance spectroscopy.
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160. Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications.
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159. Mechanistic investigation of Rh(I)-catalysed asymmetric Suzuki–Miyaura coupling with racemic allyl halides.
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157. A Bifunctional Iminophosphorane Squaramide Catalyzed Enantioselective Synthesis of Hydroquinazolines via Intramolecular Aza-Michael Addition to α,β-Unsaturated Esters.
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155. Installing the “magic methyl” – C–H methylation in synthesis.
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154. Hydrogen borrowing catalysis using 1° and 2° alcohols: Investigation and scope leading to α and β branched products.
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153. Selectivity in organocatalysis - From qualitative to quantitative predictive models.
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152. Hydrogen Borrowing Alkylation of 1,2‐Amino Alcohols in the Synthesis of Enantioenriched γ‐Aminobutyric Acids.
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151. Synthesis of legonmycins A and B, C(7a)-hydroxylated bacterial pyrrolizidines.
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150. Mass spectrometry reveals potential of β-lactams as SARS-CoV-2 M^pro inhibitors.
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149. Masked Alkyne Equivalents for the Synthesis of Mechanically Interlocked Polyynes.
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147. Single point activation of pyridines enables reductive hydroxymethylation.
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146. autodE: Automated Calculation of Reaction Energy Profiles – Application to Organic and Organometallic Reactions.
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145. Cyclic Peptides as Chemical Probes.
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144. Primary Sulfonamide Synthesis Using the Sulfinylamine Reagent N-Sulfinyl-O-(tert-butyl)hydroxylamine, t-BuONSO.
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143. Fragment-Based Identification of Ligands for Bromodomain-Containing Factor 3 of Trypanosoma Cruzi.
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142. A Single‐Stranded DNA‐Encoded Chemical Library Based on a Stereoisomeric Scaffold Enables Ligand Discovery by Modular Assembly of Building Blocks.
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141. Synthesis and Structure–Activity Relationship of Dehydrodieugenol B Neolignans against Trypanosoma cruzi.
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140. Enzymatic Kinetic Resolution by Addition of Oxygen.
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139. Inhibition of the SUV4-20 H1 histone methyltransferase increases frataxin expression in Friedreich’s ataxia patient cells.
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138. The 2‐Pyridyl Problem: Challenging Nucleophiles in Cross‐Coupling Arylations.
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137. α-Tertiary Dialkyl Ether Synthesis via Reductive Photocatalytic α-Functionalization of Alkyl Enol Ethers.
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132. Super-resolution RESOLFT microscopy of lipid bilayers using a fluorophore-switch dyad.
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130. A Modular and Divergent Approach to Spirocyclic Pyrrolidines.
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129. Synthesis of Fluorinated Alkyl Aryl Ethers by Palladium-Catalyzed C–O Cross-Coupling.
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127. Coupled metabolic cycles allow out‐of‐equilibrium autopoietic vesicle replication.
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126. Selective fragments for the CREBBP bromodomain identified from an Encoded Self‑Assembly Chemical Library.
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125. A Heck reaction/photochemical alkene isomerization sequence to prepare functionalized quinolines.
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124. Controlling gene expression with light: a multidisciplinary endeavour.
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Biochem Soc Trans, 2020, 48, 1645.

123. Synthesis of Cyclo[18]carbon via Debromination of C₁₈Br₆.
Scriven, L. M., Kaiser, K., Schulz, F., Sterling, A. J., Woltering, S. L., Gawel, P., Christensen, K. E., Anderson, H. L. and Gross, L.
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122. Atropisomerism in diarylamines: structural requirements and mechanisms of conformational interconversion.
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Angew. Chem. Int. Ed., 2020, 59, 18670.

121. Hydrogen Bonding Phase-Transfer Catalysis with Ionic Reactants: Enantioselective Synthesis of γ-Fluoroamines.
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120. Single‐molecule observation of intermediates in bioorthogonal 2‐cyanobenzothiazole chemistry.
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Angew. Chem. Int. Ed., 2020, 59, 15711.

119. BIMP Catalyzed 1,3-Prototropic Shift for the Highly Enantioselective Synthesis of Conjugated Cyclohexenones.
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118. Structure-activity relationship study of cytotoxic neolignan derivatives using multivariate analysis and computation-aided drug design.
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117. Reversible photo-control over transmembrane anion transport using visible-light responsive supramolecular carriers.
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116. Engineered anti-inflammatory peptides inspired by mapping an evasin-chemokine interaction.
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115. α‐Amidoaldehydes as substrates in rhodium‐catalyzed intermolecular alkyne hydroacylation: The synthesis of α‐amidoketones.
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114. Palladium-Catalyzed Desulfinative Cross-Couplings.
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113. Organophotochemical S_NAr Reactions of Mildly Electron‐Poor Fluoroarenes.
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112. Synthesis of All-carbon Disubstituted Bicyclo[1.1.1]pentanes by Iron-Catalyzed Kumada Cross-Coupling.
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111. Control of Absolute Stereochemistry in Transition‐Metal‐Catalyzed Hydrogen Borrowing Reactions.
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110. Consecutive 5′- and 3′-amide linkages stabilise antisense oligonucleotides and elicit an efficient RNase H response.
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109. Transmembrane anion transport mediated by halogen bonding and hydrogen bonding triazole anionophores.
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108. Rationalizing the diverse reactivity of [1.1.1]propellane through sigma-pi-delocalization.
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107. Enantiomerically Enriched Tetrahydropyridine Allyl Chlorides.
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106. An Asymmetric Suzuki–Miyaura Approach to Prostaglandins: Synthesis of Tafluprost.
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105. A hydrogen borrowing annulation strategy for the stereocontrolled synthesis of saturated aza-heterocycles.
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104. Enantioconvergent alkylation of ketones with racemic secondary alcohols via hydrogen borrowing catalysis.
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103. Double and triple ionization of isocyanic acid.
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102. Mechanistic Studies of the Palladium-Catalyzed Desulfinative Cross-Coupling of Aryl Bromides and (Hetero)Aryl Sulfinate Salts.
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101. A Modular, Enantioselective Synthesis of Resolvins D3, E1, and Hybrids.
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100. Synthesis of the cyclopentane core of pepluanin A.
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99. Chemo- and Regioselective Synthesis of Acyl-Cyclohexenes by a Tandem Acceptorless Dehydrogenation-[1,5]-Hydride Shift Cascade.
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98. [1.1.1]Propellane.
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97. α-Amino Radicals via Photocatalytic Single-Electron Reduction of Imine Derivatives.
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96. Bicyclic Lactams Derived from Serine or Cysteine and 2-Methylpropanal.
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95. Inhibitors of JmjC-Containing Histone Demethylases.
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94. ¹⁸F-Trifluoromethanesulfinate Enables Direct C–H ¹⁸F-Trifluoromethylation of Native Aromatic Residues in Peptides.
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93. Dearomative Photocatalytic Construction of Bridged 1,3-Diazepanes.
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92. Catalytic Asymmetric Suzuki–Miyaura Couplings.
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91. Structural Insights into Interaction Mechanisms of Alternative Piperazine-urea YEATS Domain Binders in MLLT1.
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90. Iridium-Catalyzed Reductive Coupling of Grignard Reagents and Tertiary Amides.
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89. Synthesis of highly fluorinated arene complexes of [Rh(chelating phosphine)]+ cations, and their use in synthesis and catalysis.
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88. ¹⁹F NMR studies on γ-butyrobetaine hydroxylase provide mechanistic insights and suggest a dual inhibition mode.
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87. How formaldehyde reacts with amino acids.
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86. Characterisation of utrophin modulator SMT C1100 as a non-competitive inhibitor of firefly luciferase.
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85. Synthesis of Cyclic Alkenyl Dimethylsiloxanes from Alkynyl Benzyldimethylsilanes and Application in Polyene Synthesis
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84. Convergent Total Syntheses of (−)‐Rubriflordilactone B and (−)‐pseudo‐Rubriflordilactone B
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83. Highly enantioselective rhodium-catalyzed cross-coupling of boronic acids and racemic allyl halides.
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82. A General Route to Bicyclo[1.1.1]pentanes through Photoredox Catalysis
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81. Desymmetrization of Meso-bisphosphates via Rhodium Catalyzed Asymmetric Allylic Arylation
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80. Bicyclic Boronate VNRX-5133 Inhibits Metallo- and Serine-β-Lactamases
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79. Modular Sulfondiimine Synthesis Using a Stable Sulfinylamine Reagent
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78. Iridium-Catalyzed Aza-Spirocyclization of Indole-Tethered Amides: An Interrupted Pictet–Spengler Reaction
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77. Retooling Asymmetric Conjugate Additions for Sterically Demanding Substrates with an Iterative Data-Driven Approach
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76. Rhodium-catalysed vinyl 1,4-conjugate addition coupled with Sharpless asymmetric dihydroxylation in the synthesis of the CDE ring fragment of pectenotoxin-4
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75. Synthesis and biophysical properties of carbamate-locked nucleic acid (LNA) oligonucleotides with potential antisense applications
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74. Intramolecular Aldol Ring Closures of Cysteine Derivatives Leading to Densely Functionalised Pyroglutamates
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73. Total Synthesis of Berkeleylactone A
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72. Dehydrodieugenol B derivatives as antiparasitic agents: Synthesis and biological activity against Trypanosoma cruzi
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71. A General Copper-Catalyzed Synthesis of Ynamides from 1,2-Dichloroenamides​
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70. A halogen-bonding foldamer molecular film for selective reagentless anion sensing in water
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69. Synthesis of Enantioenriched α‐Chiral Bicyclo[1.1.1]pentane​​
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68. A chemically fuelled self-replicator
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67. Practical and scalable kinetic resolution of BINOLs mediated by a chiral counterion
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66. Dithiane-Directed Rh(III)-Catalyzed Amidation of Unactivated C(sp3)-H Bonds
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65. The fluorination of C–H bonds: developments and perspectives​
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64. Primary α-Tertiary Amine Synthesis via α-C–H Functionalization
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63. Anion recognition in water by charge-neutral halogen and chalcogen bonding foldamer receptors​
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62. Chemical Probes​
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61. Hydrogen Bonding Phase-Transfer Catalysis with Potassium Fluoride: Enantioselective Synthesis of β-Fluoroamines
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60. Conformational Effects on Physical-Organic Descriptors – the Case of Sterimol Steric Parameters​
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59. Hydrogen bond enabled dynamic kinetic resolution of axially chiral amides mediated by a chiral counterion
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58. Chemical epigenetics: the impact of chemical‐ and chemical biology techniques on bromodomain target validation​
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57. Desymmetrization of meso-bisphosphates using copper catalysis and alkylzirconocene nucleophiles
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56. Data-mining the diaryl(thio)urea conformational landscape: Understanding the contrasting behavior of ureas and thioureas with quantum chemistry
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55. Non‐Hydrolytic β‐Lactam Antibiotic Fragmentation by L,D‐Transpeptidases and Serine β‐Lactamase Cysteine Variants
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54. Enantioselective rhodium-catalysed insertion of trifluorodiazoethanes into tin hydrides
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53. Design, Synthesis and Characterization of Covalent KDM5 Inhibitors
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52. A structure-based approach towards identification of inhibitory fragments for eleven-nineteen-leukemia protein (ENL)
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51. Target Identification Using Chemical Probes​
Moustakim, M., Ling Felce, S., Zaarour, N., Farnie, G., McCann, F. E. and Brennan, P. E.
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50. Stereospecific 1,3-H Transfer of Indenols Proceeds via Persistent Ion-Pairs Anchored By NH···Pi Interactions
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49. Copper-catalysed synthesis of alkylidene 2-pyrrolinone derivatives from the combination of α-keto amides and alkynes
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48. Discovery of an MLLT1/3 YEATS Domain Chemical Probe
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47. Enantioselective Silver-Catalyzed Cascade Synthesis of Fused Lactone and Lactam Oxazolines
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46. Post-translational site-selective protein backbone α-deuteration
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45. Principles and Applications of Fragment-based Drug Discovery for Chemical Probes
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44. Bifunctional Iminophosphorane Catalysed Enantioselective Sulfa-Michael Addition of Alkyl Thiols to Alkenyl Benzimidazoles
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43. Photocatalytic Reverse Polarity Povarov Reaction
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42. Polyyne formation via skeletal rearrangement induced by atomic manipulation
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41. A Bench-Stable Transfer Reagent for the Synthesis of Trifluoromethyl-sulfonimidamides from Sulfinamides
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40. A transient self-assembling self-replicator
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39. The Plant Cysteine Oxidases from Arabidopsis thaliana are kinetically tailored to act as oxygen sensors
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38. Roles of 2-oxoglutarate oxygenases and isopenicillin N synthase in β-lactam biosynthesis
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37. Synthesis and Applications of Highly Functionalized 1-Halo-3-Substituted Bicyclo[1.1.1]pentanes
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36. Rh(DPEPhos)-Catalyzed Alkyne Hydroacylation using β-Carbonyl Substituted Aldehydes. Mechanistic Insight Leads to Low Catalyst Loadings that Enables Selective Catalysis on Gram-Scale
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35. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability
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Bioorg. Med. Chem., 2018, 26, 2937.

34. Asymmetric nucleophilic fluorination under hydrogen bonding phase-transfer catalysis
Ascough, D. M. H., Pupo, G., Ibba, F., Vicini, A. C., Ricci, P., Christensen, K. E., Pfeifer, L. Morphy, J. R., Brown, J. M., Paton, R. S. and Gouverneur, V.
Science, 2018, 360, 638.

33. An enamine controlling group for rhodium-catalyzed intermolecular hydroacylation
Straker, R. N., Formica, M., Lupton, J. D., Niu, J. and Willis, M. C.
Tetrahedron, 2018, 74, 5408.

32. Discovery of a novel allosteric inhibitor scaffold for polyadenosine-diphosphate-ribose polymerase 14 (PARP14) macrodomain 2
Moustakim, M., Riedel, K., Schuller, M., Gehring, A. P., Monteiro, O. P., Martin, S. P., Fedorov, O., Heer, J., Dixon, D. J., Elkins, J. M., Knapp, S., Bracher, F. and Brennan, P. E.
Bioorg. Med. Chem., 2018, 26, 2965.

31. Molecular machines for catalysis
van Dijk, L., Tilby, M. J., Szpera, R., Smith, O. A., Bunce, H. A. P. and Fletcher, S. P.
Nature Rev. Chem., 2018, 2, 0117.

30. Structure activity relationship studies on rhodanines and derived enethiol inhibitors of metallo-β-lactamases
Zhang, D., Markoulides, M. S., Stepanovs, D., Rydzik, A. M., El-Hussein, A., Bon, C., Kamps, J. J. A. G., Umland, K.-D., Collins, P. M., Cahill, S. T., Wanga, D. Y., von Delft, F., Brem, J., McDonough, M. A. and Schofield, C. J.
Bioorg. Med. Chem., 2018, 26, 2928.

29. Spironaphthoxazine switchable dyes for biological imaging
Xiong, Y., Vargas Jentzsch, A., Osterrieth, J. W. M., Sezgin, E., Sazanovich, I. W., Reglinski, K., Galiani, S., Parker, A. W., Eggeling, C. and Anderson, H. L.
Chem. Sci., 2018, 9, 3029.

28. Formation of quaternary centres by copper catalysed asymmetric conjugate addition to β-substituted cyclopentenones with the aid of a quantitative structure–selectivity relationship
Ardkhean, R., Mortimore, M., Paton, R. S. and Fletcher, S. P.
Chem. Sci., 2018, 9, 2628.

27. Synthesis of Polyynes Using Dicobalt Masking Groups
Kohn, D. R., Gawel, P., Xiong, Y., Christensen, K. E. and Anderson, H. L.
J. Org. Chem., 2018, 83, 2077.

26. Detecting Mechanochemical Atropisomerization within an STM Break Junction
Leary, E., Roche, C., Jiang, H., Grace, I., González, M. T., Rubio-Bollinger, G., Romero-Muñiz, C., Xiong, Y., Al-Galiby, Q., Noori, M., Lebedeva, M. A., Porfyrakis, K., Agrait, N., Hodgson, A., Higgins, S. J., Lambert, C. J., Anderson, H. L. and Nichols, R. J
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25. Total synthesis of (−)-himalensine A
Shi, H., Michaelides, I. N., Darses, B., Jakubec, P., Nguyen, Q. N. N., Paton, R. S. and Dixon, D. J.
J. Am. Chem. Soc. 2017, 139, 17755.

24. Hexafluoroisopropanol as a highly versatile solvent
Colomer, I., Chamberlain, A. E. R., Haughey, M. B., Donohoe, T. J.
Nature Rev. Chem. 2017, 1, 0088.

23. One-pot, Three-Component Sulfonimidamide Synthesis exploiting the Sulfinylamine Reagent N-Sulfinyltritylamine, TrNSO
Davies, T. Q., Hall, A. and Willis, M. C.
Angew. Chem. Int. Ed. 2017, 56, 14937.

22. Copper-Catalyzed Synthesis and Applications of Yndiamide
Mansfield, S. J., Christensen, K. E., Thompson, A. L., Ma, K., Jones, M. W., Mekareeya, A. and Anderson​, E. A.
Angew. Chem. Int. Ed. 2017, 56, 14428.

21. Enantioselective Conjugate Addition Catalyzed by a Copper Phosphoramidite Complex: Computational and Experimental Exploration of Asymmetric Induction
Ardkhean, R.,  Roth, P. M. C., Maksymowicz, R. M., Curran, A., Peng, Q., Paton, R. S. and Fletcher, S. P.
ACS Catal. 2017, 7, 6729.

20. Crotonases - Nature's Exceedingly Convertible Catalysts
Lohans, C. T., Wang, D. Y., Wang, J., Hamed, R. B., Schofield, C. J.
ACS Catal. 2017, 7, 6587.

19. Exploiting Carbonyl Groups to Control Intermolecular Rhodium-Catalyzed Alkene and Alkyne Hydroacylation
Coxon, T. J., Fernandez, M., Barwick-Silk, J., McKay, A. I., Britton, L. E., Weller, A. S., Willis, M. C.
J. Am. Chem. Soc. 2017, 139, 10142.

18. Visible light photocatalysis of 6π heterocyclization
Münster, N., Parker, N. A., van Dijk, L., Paton, R. S., Smith, M. D.
Angew. Chem. Int. Ed. 2017, 56, 9468.

17. Unexpected Interactions between Alkyl Straps and Pyridine Ligands in Sulfur-Strapped Porphyrin Nanorings
Roche, C., Lou, Q., Gil-Ramirez, G., Jiang, H.-W., Kohn, D. R., Xiong, Y., Thompson, A. L., Anderson, H. L.
J. Org. Chem. 2017, 82, 7446.

16. Potential for minimal self-replicating systems in a dynamic combinatorial library of equilibrating imines
Morrow, S. M., Bissette, A. J., Fletcher, S. P.
Tetrahedron 2017, 73, 5005.

15. Transmission of chirality through space and across length scales
Morrow, S. M., Bissette, A. J. and Fletcher, S. P.
Nature Nanotechnology 2017, 12, 410.

14. Structural and stereoelectronic insights into oxygenase-catalyzed formation of ethylene from 2-oxoglutarate
Zhang, Z., Smart, T. J., Choi, H., Hardy, F., Lohansa, C. T., Abboud, M. I., Richardson, M. S. W., Paton, R. S., McDonough, M. A. and Schofield, C. J.
Proc. Natl. Acad. Sci. 2017, 114, 4667. 

13. Neutral iodotriazole foldamers as tetradentate halogen bonding anion receptors
Borissov, A., Lim, J. Y. C., Brown, A., Christensen, K. E., Thompson, A. L., Smith, M. D. and Beer, P. D.
Chem. Commun. 2017, 53, 2483.

12. Discovery of a PCAF Bromodomain Chemical Probe
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Angew. Chem. Int. Ed. 2017, 56, 827. DOI: 10.1002/anie.201610816.

11. Umpolung synthesis of branched α-functionalized amines from imines via photocatalytic three-component reductive coupling reactions
Fuentes de Arriba, A. L., Urbitsch, F., Dixon, D. J.
Chem. Commun. 2016, 52, 14434.

10. A Cascade Strategy Enables a Total Synthesis of (+/-)-Morphine
Chu, S., Münster, N., Balan, T., Smith. M. D.
Angew. Chem. Int. Ed. 2016, 55, 14306.

9. Posttranslational mutagenesis: A chemical strategy for exploring protein side-chain diversity
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Science 2016, 354, 597.

8. Chemical Probes and Inhibitors of Bromodomains outside the BET family
Moustakim, M., Clark, P. G. K., Hay, D. A., Dixon, D. J. and Brennan, P. E.
Med. Chem. Commun. 2016, 7, 2246.

7. Photoswitchable Spiropyran Dyads for Biological Imaging
Xiong, Y., Rivera-Fuentes, P., Sezgin, E., Jentzsch, A. V., Eggeling, C. and Anderson, H. L.
Org. Lett. 2016, 8, 3666.

6. Cp₂ZrMeCl: A Reagent for Asymmetric Methyl Addition
Garrec, K. and Fletcher, S. P.
Org. Lett. 2016, 8, 3814.

5. Recent Applications in Natural Product Synthesis of Dihydrofuran and -pyran Formation by Ring-closing Alkene Metathesis
Jacques, R., Pal, R., Parker, N. A., Sear, C. E., Smith, P. W., Ribaucourt, A. and Hodgson, D. M.
Org. Biomol. Chem. 2016, 14, 5875.

4. Organocatalytic Enantioselective Desymmetrisation
Borissov, A., Davies, T. Q., Ellis, S. R., Fleming T. F., Richardson, M. S. W. and Dixon, D. J.
Chem. Soc. Rev. 2016, 45, 5474.

3. Cascade Polycyclizations in Natural Product Synthesis
Ardkhean, R., Caputo, D. F. J., Morrow, S. M., Shi H., Xiong, Y and Anderson, E. A.
Chem. Soc. Rev. 2016, 45, 1557.

2. Strategic Application and Transformation of ortho-Disubstituted Phenyl and Cyclopropyl Ketones to Expand the Scope of Hydrogen Borrowing Catalysis
Frost, J. R., Cheong, C. B., Akhtar, W. M., Caputo, D. F. J., Stevenson, N. G. and Donohoe, T. J.
J. Am. Chem. Soc. 2015, 137, 15664.

1. Active-Metal Template Synthesis of a Halogen-Bonding Rotaxane for Anion Recognition
Langton, M. J., Xiong, Y. and Beer, P. D.
Chem. Eur. J. 2015, 21, 18910.